Biochemical Assay Services

Free Choice Kinase Assay Projects / Kinase Assays

Field of Application

Free choice kinase assay projects allow characterization of your test compounds in a total flexible mode. For each project you can freely define (i) the number of kinase assays, (ii) the number of test compounds (iii) and the number of data points for each test compound (i.e. number of concentrations and replicates). All kinase assays are designed to measure biochemical kinase activity.

Our Products

Number Kinase Synonyms
1 ABL1 E255K ABL1, c-Abl, JTK7, p150
2 ABL1 F317I ABL1, ABL, JTK7, p150, c-ABL, v-abl
3 ABL1 G250E ABL1, ABL, JTK7, p150, c-ABL, v-abl
4 ABL1 H396P ABL1, ABL, JTK7, p150, c-ABL, v-abl
5 ABL1 M351T ABL1, ABL, JTK7, p150, c-ABL, v-abl
6 ABL1 Q252H ABL1, ABL, JTK7, p150, c-ABL, v-abl
7 ABL1 T315I ABL1, ABL, JTK7, p150, c-ABL, v-abl
8 ABL1 wt ABL1, ABL, JTK7, p150, c-ABL, v-abl
9 ABL1 Y253F ABL1, ABL, JTK7, p150, c-ABL, v-abl
10 ABL2 ABL2, ABLL, ARG
11 ACK1 TNK2, ACK, p21cdc42Hs, Activated CDC42 kinase 1
12 ACV-R1 ACVR1, ACTRI, ACVRLK2, ALK2, SKR1
13 ACV-R1B ACVR1B, ACTRIB, ACVRLK4, ALK4, SKR2
14 ACV-R2A ACVR2, ACTRII
15 ACV-R2B ActR-IIB, ACTRIIB
16 ACV-RL1 ACVRL1, ACVRLK1, ALK-1, ALK1, HHT, HHT2, ORW2, SKR3
17 AKT1 aa1-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
18 AKT1 aa106-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
19 AKT2 aa1-481 AKT2, PKBB, PKBBETA, PKB beta, PRKBB, RAC-beta, RAC-PK-beta
20 AKT2 aa107-481 AKT2, PRKBB, PKBBETA, RAC-BETA
21 AKT3 aa1-479 AKT3, PKBG, PKB gamma, PRKBG, RAC-gamma, RAC-PK-gamma, STK-2, DKFZp434N0250
22 AKT3 aa106-479 AKT3, PKBG, PRKBG, STK-2, RAC-gamma, RAC-PK-gamma
23 ALK C1156Y (GST-HIS-tag) ALK, CD246, NBLST3
24 ALK F1174L (GST-HIS-tag) ALK, CD246, NBLST3
25 ALK F1174S (GST-HIS-tag) ALK, CD246, NBLST3
26 ALK G1202R (GST-HIS-tag) ALK, CD246, NBLST3
27 ALK L1196M (GST-HIS-tag) ALK, CD246, NBLST3
28 ALK R1275Q (GST-HIS-tag) ALK, CD246, NBLST3
29 ALK wt (GST-HIS-tag) ALK, CD246, NBLST3
30 AMPK-alpha1 aa1-550 PRKAA1, MGC33776, MGC57364
31 ARK5 NUAK1, KIAA0537
32 ASK1 MAP3K5, ASK1, MAPKKK5, MEKK5
33 Aurora-A AURKA, AIK, ARK1, AURA, BTAK, STK15, MGC34538, STK6
34 Aurora-B AURKB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AIM-1, STK12
35 Aurora-C AURKC, AIE2, AIK3, STK13
36 AXL AXL, EC, UFO
37 B-RAF V600E BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
38 B-RAF wt BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
39 BLK BLK, n/a
40 BMPR1A BMPR1A, ACVRLK3, ALK3
41 BMPR1B BMPR1B, ALK6, CDw293
42 BMX BMX, ETK, PSCTK2, PSCTK3
43 BRK PTK6, n/a
44 BRSK1 BRSK1, KIAA1811
45 BRSK2 C11orf7, FLJ41362, HUSSY-12, PEN11B, SAD1, STK29
46 BTK BTK, AGMX1, AT, ATK, BPK, PSCTK1
47 BUB1B BUB1B, BUBR1, Bub1A, MAD3L, hBUBR1
48 CAMK1D CAMK1D, CKLiK, CaM-K1, CaMKID
49 CAMK2A CAMK2A, CAMKA, KIAA0968
50 CAMK2B CAMK2B, CAM2, CAMK2, CAMKB, MGC29528
51 CAMK2D CAMK2D, CAMKD, MGC44911, CaMKII delta
52 CAMK2G CAMK2G, CAMK, CAMK-II, CAMKG, MGC26678
53 CAMK4 CAMK4, CaMK-GR, MGC36771
54 CAMKK1 CAMKK1, CAMKKA, DKFZp761M0423, MGC34095
55 CAMKK2 CAMKK2, CAMKK, CAMKKB, KIAA0787, MGC15254
56 CCDC6-RET CCDC6-RET, CCDC6-RETa
57 CDC42BPA CDC42BPA, MRCK-alpha
58 CDC42BPB CDC42BPB, MRCK-beta, MRCKb
59 CDC7/DBF4 CDC7, CDC7L1, HsCdc7, HsCDC7, Hsk1, huCdc7
60 CDK1/CycA2 CDC2, p34
61 CDK1/CycB1 CDC2, p34
62 CDK1/CycE1 CDC2, p34
63 CDK12 R722C/CycK CDK12, CRKRS, CRK7
64 CDK12 wt/CycK CDK12, CRKRS, CRK7
65 CDK13/CycK CDK13, CDC2L, CDC2L5, CHED
66 CDK16/CycY CDK16, PCTAIRE1, PCTAIRE, PCTGAIRE, PCTK1
67 CDK17/p35NCK CDK17, PCTAIRE2, PCTK2
68 CDK18/CycY CDK18, PCTAIRE, PCTAIRE3, PCTK3
69 CDK19/CycC CDK19, CDC2L6, CDK11
70 CDK2/CycA2 CDK2, p33(CDK2)
71 CDK2/CycD1 CDK2, p33
72 CDK2/CycE1 CDK2, p33(CDK2)
73 CDK20/CycH CDK20, CAK-kinase p42
74 CDK20/CycT1 CDK20, CAK-kinase p42, CCRK, CDCH, p42, PNQALRE
75 CDK3/CycC CDK3, CDKN3
76 CDK3/CycE1 CDK3, n/a
77 CDK4/CycD1 CDK4, CMM3, PSK-J3, MGC14458
78 CDK4/CycD2 CDK4, CMM3, PSK-J3
79 CDK4/CycD3 CDK4, CMM3, PSK-J3, MGC14458
80 CDK5/p25NCK CDK5, PSSALRE
81 CDK5/p35NCK CDK5, PSSALRE
82 CDK6/CycD1 CDK6, PLSTIRE, MGC59692
83 CDK6/CycD2 CDK6, PLSTIRE
84 CDK6/CycD3 CDK6, PLSTIRE
85 CDK7/CycH/MAT1 CDK7, CAK1, CDKN7, STK1, p39MO15
86 CDK8/CycC CDK8, K35
87 CDK9/CycK CDK9, C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase
88 CDK9/CycT1 CDK9, C-2k, CDC2L4K35, PITALRE, TAK
89 CHK1 CHEK1, n/a
90 CHK2 CHEK2, CDS1, HuCds1, PP1425, RAD53, bA444G7
91 CK1-alpha1 CSNK1A1, CK1, HLCDGP1, PRO2975
92 CK1-delta CSNK1D, HCKID
93 CK1-epsilon CSNK1E, CKIe, HCKIE, MGC10398
94 CK1-gamma1 CSNK1G1
95 CK1-gamma2 CSNK1G2, CK1g2
96 CK1-gamma3 CSNK1G3
97 CK2-alpha1 CSNK2A1, CKII, CK2A1
98 CK2-alpha2 CSNK2A2, n/a
99 CLK1 CLK1, CLK, CLK/STY
100 CLK2 CLK2, MGC61500, clk2, hCLK2
101 CLK3 CLK3, PHCLK3, PHCLK3/152
102 CLK4 CLK4, DKFZp686A20267, CDC-like kinase 4
103 COT MAP3K8, EST, ESTF, TPL2, Tpl-2, c-COT
104 CSF1-R CSF1R, C-FMS, CD115, CSF-1-R, CSFR, FIM2, FMS
105 CSK CSK, n/a
106 DAPK1 DAPK1, n/a
107 DAPK2 DAPK2, DRP-1
108 DAPK3 DAPK3, ZIP, ZIPK
109 DCAMKL2 DCLK2, DCLK, KIAA0369
110 DDR2 N456S DDR2, MIG20a, NTRKR3, TKT, TYRO10
111 DDR2 T654M DDR2, MIG20a, NTRKR3, TKT, TYRO10
112 DDR2 wt DDR2, MIG20a, NTRKR3, TKT, TYRO10
113 DMPK DMPK, DM, DM1, DM1PK, DMK
114 DNA-PK PRKDC, DNAPK, DNPK1, HYRC, HYRC1, XRCC7, p350
115 DYRK1A DYRK1A, DYRK, DYRK1, HP86, MNB, MNBH
116 DYRK1B DYRK1B, MIRK
117 DYRK2 DYRK2
118 DYRK3 DYRK3, DYRK5, RED, REDK
119 DYRK4 DYRK4
120 EEF2K EEF2K, HSU93850, MGC45041, eEF-2K
121 EGF-R C797S EGF-R, ERBB, ERBB1
122 EGF-R d746-750 EGFR, ERBB, mENA, ERBB1
123 EGF-R d747-749/A750P EGFR, ERBB, mENA, ERBB1
124 EGF-R d747-752/P753S EGFR, ERBB, mENA, ERBB1
125 EGF-R d752-759 EGFR, ERBB, mENA, ERBB1
126 EGF-R G719C EGFR, ERBB, mENA, ERBB1
127 EGF-R G719S EGFR, ERBB, mENA, ERBB1
128 EGF-R L858R EGFR, ERBB, ERBB1
129 EGF-R L861Q EGFR, ERBB, mENA, ERBB1
130 EGF-R T790M EGFR, ERBB, ERBB1
131 EGF-R T790M/L858R EGFR, ERBB, ERBB1
132 EGF-R wt EGFR, ERBB, mENA, ERBB1
133 EIF2AK2 EIF2AK2, EIF2AK1, PKR, PRKR
134 EIF2AK3 EIF2AK3, DKFZp781H1925, PEK, PERK, WRS
135 EML4 ALK ALK
136 EML4 ALK F1174L ALK
137 EPHA1 EPHA1, EPH, EPHT, EPHT1
138 EPHA2 EPHA2, ECK
139 EPHA3 EPHA3, ETK, ETK1, EphA3, HEKECK, HEK4, TYRO4
140 EPHA4 EPHA4, HEK8, SEK, TYRO1
141 EPHA5 EPHA5, CEK7, EHK1, EphA5, HEK7, Hek7, TYRO4
142 EPHA6 EPHA6, EHK2, EHK-2, EPA6
143 EPHA7 EPHA7, EHK3, HEK11
144 EPHA8 EPHA8, EEK, EphA8, HEK3, KIAA1459
145 EPHB1 EPHB1, ELK, NET, Hek6, EPHT2
146 EPHB2 EPHB2, DRT, ERK, Hek5, EPHT3, Tyro5
147 EPHB3 EPHB3, ETK2, HEK2, TYRO6
148 EPHB4 EPHB4, HTK, MYK1, TYRO11
149 ERBB2 775YVMA776 ERBB2, CD340, HER2, MLN19, NGL, TKR1
150 ERBB2 wt ERBB2, NEU, NGL, HER2, TKR1, HER-2
151 ERBB4 ERBB4, n/a
152 ERK1 MAPK3, ERT2, HS44KDAP, HUMKER1A, P44ERK1, P44MAPK, PRKM3
153 ERK2 MAPK1, ERK, ERT1, MAPK2, P42MAPK, PRKM1, PRKM2, p38, p40, p41
154 ERK5 MAPK7, BMK1, ERK4, PRKM7
155 ERK7 MAPK15, ERK8, MAPK15
156 FAK aa2-1052 PTK2, FADK, pp125FAK
157 FER FER, TYK3, c-FER, p94-FER
158 FES FES, FPS
159 FGF-R1 V561M FGFR1, FGFR-1, bFGF-R, FLT2, CEK, CD331
160 FGF-R1 wt FGFR1, H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM
161 FGF-R2 FGFR2, FGFR2, BEK, BFR-1, CD332, CEK3, CFD1, ECT1, FGFR-2, JWS, KGFR, KSAM, K-SAM, TK14, TK25
162 FGF-R3 G697C FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
163 FGF-R3 K650E FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
164 FGF-R3 K650M FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
165 FGF-R3 wt FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
166 FGF-R4 FGFR4, TKF, JTK2, MGC20292
167 FGR FGR, SRC2, c-fgr, p55c-fgr
168 FLT3 D835Y FLT3, CD135, FLK2, STK-1, STK1
169 FLT3 ITD FLT3, CD135, FLK2, STK-1, STK1
170 FLT3 wt FLT3, CD135, FLK2, STK-1, STK1
171 FRK FRK, GTK, PTK5, RAK
172 FYN wt FYN, SLK, SYN, p59-Fyn
173 FYN Y531F FYN, SLK, SYN, p59-FYN, cFYN
174 GRK2 ADRBK1
175 GRK3 ADRBK2
176 GRK4 GRK4, GPRK2L, GPRK4, GRK4a, IT11
177 GRK5 GRK5
178 GRK6 GRK6
179 GRK7 GRK7
180 GSG2 GSG2, Haspin
181 GSK3-alpha GSK3A
182 GSK3-beta GSK3B
183 HCK HCK, JTK9
184 HIPK1 HIPK1, KIAA0630, MGC26642, MGC33446, MGC33548, Myak, Nbak2
185 HIPK2 HIPK2, PRO0593
186 HIPK3 HIPK3, ANPK, DYRK6, FIST, FIST3, PKY, YAK1
187 HIPK4 HIPK4, FLJ32818
188 HRI EIF2AK1, HCR
189 IGF1-R IGF1R, JTK13
190 IKK-alpha CHUK, IKBKA, IKK1, IKKA, NFKBIKA, TCF16
191 IKK-beta IKBKB, IKK2, IKKB, NFKBIKB
192 IKK-epsilon IKBKE, IKKE, IKKI, IKK-i, KIAA0151
193 INS-R INSR, n/a
194 INSR-R INSRR, IRR
195 IRAK1 IRAK1, IRAK, Pelle
196 IRAK4 (untagged) IRAK4, REN64, NY-REN-64
197 ITK ITK, EMT 2, LYK 2, PSCTK2 2, IL2-inducible T-cell kinase
198 JAK1 aa583-1154 S729C JAK1, JAK1A, JAK1B, JTK3
199 JAK1 aa583-1154 wt JAK1, JAK1A, JAK1B, JTK3
200 JAK2 JAK2, n/a
201 JAK3 JAK3, JAKL, L-JAK, LJAK
202 JNK1 MAPK8, PRKM8, SAPK1, JNK1-alpha1
203 JNK2 MAPK9, PRKM9, p54aSAPK, JNK2-alpha2
204 JNK3 MAPK10, JNK3A, p54bSAPK
205 KIT A829P KIT, C-Kit, PBT, CD117, SCFR, c-kit
206 KIT D816H KIT, C-Kit, PBT, CD117, SCFR, c-kit
207 KIT D816V KIT, C-Kit, PBT, CD117, SCFR, c-kit
208 KIT T670I KIT, CD117, SCFR, PBT, C-Kit
209 KIT V559D KIT, C-Kit, PBT, CD117, SCFR, c-kit
210 KIT V559D/T670I KIT, C-Kit, PBT, CD117, SCFR, c-kit
211 KIT V559D/V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
212 KIT V560G KIT, C-Kit, PBT, CD117, SCFR, c-kit
213 KIT V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
214 KIT wt KIT, C-Kit, PBT, CD117, SCFR, c-kit
215 LCK LCK, n/a
216 LIMK1 LIMK1, LIMK
217 LIMK2 LIMK2
218 LRRK2 G2019S LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
219 LRRK2 I2020T LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
220 LRRK2 R1441C LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
221 LRRK2 wt LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
222 LTK LTK, TYK1
223 LYN LYN, JTK8
224 MAP3K1 MAP3K1, MAPKKK1, MEKK, MEKK1
225 MAP3K10 MAP3K10, MLK2, MST, MEKK10
226 MAP3K11 MAP3K11, MGC17114, MLK-3, PTK1, SPRK
227 MAP3K7/MAP3K7IP1 MAP3K7, TAK1, TGF1a, MEKK7
228 MAP3K9 MAP3K9, MLK1, PRKE1, MEKK9
229 MAP4K2 MAP4K2, BL44, GCK, RAB8IP
230 MAP4K4 MAP4K4, HGK, MEKKK4, NIK
231 MAP4K5 MAP4K5, KHS1, GCKR, KHS, MAPKKKK5
232 MAPKAPK2 MAPKAPK2, n/a
233 MAPKAPK3 MAPKAPK3, 3PK, MAPKAP, MAPKAP3
234 MAPKAPK5 MAPKAPK5, PRAK
235 MARK1 MARK1, KIAA1477
236 MARK2 MARK2, EMK1, MGC99619, PAR-1, ELKL motif kinase 1
237 MARK3 MARK3, CTAK1, KP78, PAR1A
238 MARK4 MARK4, KIAA1860, MARKL1
239 MASTL MASTL, GLW, GREATWALL, GWL, hGWL, MAST-L, THC2
240 MATK MATK, CHK, CTK, DKFZp434N1212, HHYLTK, HYL, Lsk, MGC1708, MGC2101
241 MEK1 F53L MAP2K1, MAP2K1, MAPKK1, MAPKK 1, MKK1, PRKMK1
242 MEK1 wt MAP2K1, MAPKK1, MKK1, PRKMK1
243 MEK2 MAP2K2, MAPKK2, MKK2, PRKMK2
244 MEK5 MAP2K5, MAP2K5, MAPKK5, MKK5, PRKMK5
245 MEKK2 MAP3K2, MAPKKK2, MEKK2B
246 MEKK3 MAP3K3, MAPKKK3, MEK kinase3
247 MELK MELK, PK38
248 MERTK MERTK, MER, MER-PEN, RP38
249 MET D1228H MET, HGFR, RCCP2
250 MET D1228N MET, HGFR, RCCP2
251 MET F1200I MET, HGFR, RCCP2
252 MET G1163R MET, HGFR, RCCP2
253 MET L1195V MET, HGFR, RCCP2
254 MET M1250T MET, HGFR, RCCP2
255 MET wt MET, HGFR, RCCP2
256 MET Y1230A MET, HGFR, RCCP2
257 MET Y1230C MET, HGFR, RCCP2
258 MET Y1230D MET, HGFR, RCCP2
259 MET Y1230H MET, HGFR, RCCP2
260 MET Y1235D MET, HGFR, RCCP2
261 MINK1 MINK1, B55, YSK2, MAP4K6, ZC3
262 MKK4 MAP2K4, JNKK, JNKK1, MAPKK4, MEK4, PRKMK4, SEK, SERK1
263 MKK6 S207D/T211D MAP2K6, MAPKK6, MEK6, MKK6, PRKMK6, SAPKK3
264 MKK7 MAP2K7, MAPKK7, MEK7, PRKMK7
265 MKNK1 MKNK1, MNK1
266 MKNK2 MKNK2, MNK2, GPRK7
267 MLK4 n/a, KIAA1804
268 MST1 STK4, KRS2, YSK3
269 MST2 STK3, MST-2, KRS1
270 MST3 STK24, MST-3, MST3B, STK3
271 MST4 MST4, MASK
272 mTOR FRAP1, FRAP, FRAP2, RAFT1, RAPT1, rapamycin target protein
273 MUSK MUSK, n/a
274 MYLK MYLK, smMLCK, FLJ12216, KRP, MLCK, MLCK108, MLCK210
275 MYLK2 MYLK2, KMLC, MLCK, skMLCK
276 MYLK3 MYLK3, caMLCK, MLCK2, MYLK2
277 NEK1 NEK1, NY-REN-55
278 NEK11 NEK11, FLJ23495
279 NEK2 NEK2, NLK1, HsPK21, HsPK 21
280 NEK3 NEK3, HSPK36, MGC29949
281 NEK4 NEK4, NRK2, STK2
282 NEK6 NEK6, SID6-1512
283 NEK7 NEK7, n/a
284 NEK9 NEK9, DKFZp434D0935, MGC16714, NERCC, NERCC1, Nek8
285 NIK MAP3K14, FTDCR1B, HS, HSNIK
286 NLK NLK, n/a
287 NPM1 ALK n/a, n/a
288 NPM1 ALK F1174L n/a, n/a
289 p38-alpha MAPK14, p38-alpha
290 p38-beta MAPK11, p38-beta
291 p38-delta MAPK13, n/a
292 p38-gamma MAPK12, ERK-6, ERK3, ERK5, ERK6, PRKM12, SAPK-3, SAPK3
293 PAK1 PAK1, PAKalpha
294 PAK2 PAK2, PAK65, PAKgamma
295 PAK3 PAK3, CDKN1A, MRX30, OPHN3, PAK3beta, bPAK, hPAK3
296 PAK4 PAK4, n/a
297 PAK6 PAK6, PAK5
298 PAK7 PAK7, KIAA1264, MGC26232
299 PASK PASK, DKFZP434O051, DKFZp686P2031, KIAA0135, PASKIN, STK3
300 PBK PBK, TOPK, SPK, Nori-3, FLJ14385
301 PDGFR-alpha D842V PDGFRA, PDGFR2, CD140a
302 PDGFR-alpha T674I PDGFRA, PDGFR2, CD140a
303 PDGFR-alpha V561D PDGFRA, PDGFR2, CD140a
304 PDGFR-alpha wt PDGFRA, PDGFR2, CD140a
305 PDGFR-beta PDGFRB, JTK12, PDGFR, CD140B, PDGFR1, PDGF-R-beta
306 PDK1 PDPK1, PKB-like
307 PHKG1 PHKG1, PHKg1
308 PHKG2 PHKG2, PHKg2
309 PI4K2A PI4K2A, PI4KII, PIK42A, RP11-548K23.6
310 PI4K2B PI4K2B, PI4KIIB, PI4KII-BETA, PIK42B
311 PI4KB PI4KB, NPIK, pi4K92, PI4K92, PI4Kbeta, PI4KBETA, PI4K-beta, PI4K-BETA, PI4KIIIBETA, PIK4CB
312 PIK3C2A PIK3C2A, CPK, MGC142218, PI3-K-C2A
313 PIK3C2B PIK3C2B, C2-PI3K, PI3K-C2beta
314 PIK3C2G PIK3C2G, PI3K-C2GAMMA, PI3K-C2-gamma
315 PIK3C3 PIK3C3, hVps34, MGC61518, PI3-kinase type 3, PI3K type 3, Vps34, VPS34
316 PIK3CA/PIK3R1 PIK3CA, MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha
317 PIK3CB D1067A/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
318 PIK3CB D1067V/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
319 PIK3CB D1067Y/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
320 PIK3CB E1051K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
321 PIK3CB E633K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
322 PIK3CB L1049R/PIK3R1 PIK3CB
323 PIK3CB wt/PIK3R1 PIK3CB, PI3K, PI3KBETA, PI3K-beta, PIK3C1, p110-beta
324 PIK3CD/PIK3R1 PIK3CD, p110D, P110DELTA, PI3K, PI3K-delta, p110-delta
325 PIK3CG PIK3CG, p120-PI3K, PI3CG, PI3K, PI3Kgamma, PI3K-gamma, p110-gamma
326 PIM1 PIM1, PIM
327 PIM2 PIM2, n/a
328 PIM3 PIM3, n/a
329 PIP5K1A PIP5K1A, PIP5K1-alpha, PIP5KIalpha, PtdIns(4)P-5-kinase 1 alpha
330 PIP5K1B PIP5K1B, MSS4, PIP5K1-beta, STM7
331 PIP5K1C PIP5K1C, PIP5K1-gamma, PIP5Kgamma, PIP5K-GAMMA, PIPKIg_v4
332 PKA PRKACA, MGC48865, PKA
333 PKC-alpha PRKCA, PKCA, PRKACA, PKC-alpha
334 PKC-beta1 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
335 PKC-beta2 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
336 PKC-delta PRKCD, MAY1, MGC49908, nPKC-delta
337 PKC-epsilon PRKCE, PKCE, nPKC-epsilon
338 PKC-eta PRKCH, PKC-L, PKCL, PRKCL, nPKC-eta
339 PKC-gamma PRKCG, PKCC, PKCG, SCA14, MGC57564
340 PKC-iota PRKCI, PKCI, DXS1179E, MGC26534, nPKC-iota
341 PKC-mu PRKD1, PKD, PKCM, PKC-MU
342 PKC-nu PRKD3, EPK2
343 PKC-theta PRKCQ, PRKCT, nPKC-theta
344 PKC-zeta PRKCZ, PKC2
345 PKC-zeta wt aa184-592 (PKM-zeta) PRKCZ, PKM-zeta, nPKC-zeta, PKC2
346 PKMYT1 PKMYT1, MYT1
347 PKN3 PKN3, PKNbeta, RP11-545E17.1
348 PLK1 PLK1, PLK, STPK13
349 PLK3 PLK3, CNK, FNK, PRK
350 PRK1 PKN1, DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204
351 PRK2 PKN2, PRKCL2, PAK-2
352 PRKD2 PRKD2, PKD2, HSPC187
353 PRKG1 PRKG1, PKG1, CGKI, MGC71944, PGK, PRKG1B, PRKGR1B, cGKIBETA, cGKI-alph
354 PRKG2 PRKG2, PKG2, PRKGR2, cGKII
355 PRKX PRKX, PKX1
356 PYK2 PTK2B, CADTK, CAKB, FADK2, FAK2, PKB, PTK, PYK2, RAFTK, CAK beta
357 RAF1 Y340D/Y341D (untagged) RAF1, c-RAF
358 RET E762Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
359 RET G691S RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
360 RET M918T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
361 RET R749T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
362 RET R813Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
363 RET S891A RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
364 RET V804E RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
365 RET V804L RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
366 RET V804M RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
367 RET wt RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
368 RET Y791F RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
369 RET Y806H RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
370 RIPK2 RIPK2, CARD3, CARDIAK, CCK, GIG30, RICK, RIP-2, RIP2
371 RIPK4 RIPK4, ANKK2, ANKRD3, DIK, MGC129992, MGC129993, PKK, RIP4
372 RIPK5 DSTYK, SgK496, SHIK
373 ROCK1 ROCK1, P160ROCK
374 ROCK2 ROCK2, KIAA0619, ROC2
375 RON MST1R, CD136, CDw136, PTK8
376 ROS ROS1, MCF3
377 RPS6KA1 RPS6KA1, RSK3, HU-1, MAPKAPK1A, RSK, RSK1
378 RPS6KA2 RPS6KA2, RSK1, HU-2, MAPKAPK1C, RSK, RSK3
379 RPS6KA3 RPS6KA3, HU-2, HU-3, ISPK-1, MAPKAPK1B, MRX19, RSK, RSK2
380 RPS6KA4 RPS6KA4, MSK2, RSK-B
381 RPS6KA5 RPS6KA5, MSK1, EC 2.7.11, MGC1911, MSPK1, RLPK, RSKL
382 RPS6KA6 RPS6KA6, RSK4
383 S6K RPS6KB1, S6K1, STK14A
384 S6K-beta RPS6KB2, KLS, P70-beta-1, P70-beta-2, S6K-beta2, S6K2, SRK, p70S6Kb
385 SAK PLK4, SAK, STK18
386 SGK1 SGK, n/a
387 SGK2 SGK2, H-SGK2, dJ138B7.2
388 SGK3 SGKL, CISK, SGK2, SGK3
389 SIK1 SIK1, MSK, SNF1LK, SIK, SIK-1, SNF1LK
390 SIK2 SIK2, QIK, SNF1LK2
391 SIK3 SIK3, L19, QSK, SIK-3
392 SLK SLK, KIAA0204, STK2, bA16H23.1, se20-9
393 SNARK NUAK2, DKFZp434J037
394 SNK PLK2, SNK
395 SRC (GST-HIS-tag) SRC, ASV, SRC1, c-SRC, p60-Src
396 SRMS SRMS, C20orf148, SRM, dJ697K14.1
397 SRPK1 SRPK1, SFRSK1
398 SRPK2 SRPK2, SFRSK2
399 STK17A STK17A, DRAK1
400 STK23 SRPK3, MSSK1, MGC102944
401 STK25 STK25, DKFZp686J1430, SOK1, YSK1
402 STK33 STK33
403 STK39 STK39, STLK3, DCHT, SPAK
404 SYK aa1-635 SYK, n/a
405 TAOK2 TAOK2, KIAA0881, MAP3K17, PSK, PSK1, TAO1, TAO2
406 TAOK3 TAOK3, DPK, JIK, MAP3K18, TAO kinase 3
407 TBK1 TBK1, CDC37, HSPCA, HSPCB, IKBKG, NAK, T2K, TANK, TRAF2
408 TEC TEC, PSCTK4
409 TGFB-R1 TGFBR1, ALK5, ACVRLK4
410 TGFB-R2 TGFBR2, HNPCC6, MFS2, RIIC, TGFR-2, TGFbeta-RII
411 TIE2 R849W TEK, VMCM, TIE-2, VMCM1, CD202B
412 TIE2 wt TEK, VMCM, TIE-2, VMCM1, CD202B
413 TIE2 Y1108F TEK, VMCM, TIE-2, VMCM1, CD202B
414 TIE2 Y897S TEK, VMCM, TIE-2, VMCM1, CD202B
415 TLK1 TLK1, PKU-beta, KIAA0137
416 TLK2 TLK2, MGC44450, PKU-ALPHA
417 TNK1 TNK1, n/a
418 TRK-A G667C MTC, TRK1, TRKA
419 TRK-A wt NTRK1, MTC, TRK, TRK1, TRKA
420 TRK-B NTRK2, GP145-TrkB, TRKB, Trk-B
421 TRK-C NTRK3, GP145-TrkC, TRKC, Trk-C
422 TSF1 STK16, KRCT, MPSK, PKL12
423 TSK2 TSSK2, DGS-G, SPOGA2, FLJ38613
424 TSSK1 TSSK1, FKSG81, SPOGA4, STK22D
425 TTBK1 aa1-1321 TTBK1, BDTK
426 TTBK1 aa1-480 TTBK1, BDTK
427 TTBK2 TTBK2, BDTK, KIAA1855, RP3-330M21.4
428 TTK TTK, ESK, MPS1L1, PYT
429 TXK TXK, BTKL, PSCTK5, PTK4, RLK
430 TYK2 TYK2, JTK1
431 TYRO3 TYRO3, BYK, Brt, Dtk, Sky, Tif
432 ULK2 ULK2, ATG1B, KIAA0623, Unc51.2
433 VEGF-R1 FLT1, FLT, VEGFR1
434 VEGF-R2 KDR, FLK1, VEGFR, VEGFR2
435 VEGF-R3 FLT4, PCL, VEGFR3
436 VRK1 VRK1, n/a
437 VRK2 VRK2, n/a
438 WEE1 WEE1, WEE1hu
439 WNK1 WNK1, KDP, KIAA0344, PHA2C, PRKWNK1
440 WNK2 WNK2, KIAA1760, NY-CO-43, P/OKcl.13, PRKWNK2, SDCCAG43
441 WNK3 WNK3, KIAA1566, PRKWNK3
442 YES YES, C-YES, HsT441, P61-YES
443 ZAK MLTK, mlklak, AZK
444 ZAP70 ZAP70, SRK, STD, TZK, ZAP-70

Info in Brief

Kinase Panel

444 kinases, including 91 disease-relevant kinase
mutants and 20 lipid kinases

Assay Technologies

Protein kinases: FlashPlate™-based radiometric assay;
lipid kinases: ADP-Glo™ assay technology (Promega)

ATP conc

App. ATP-Km for each kinase

Testing Modes

Single concentration measurement or IC50 profiling
(10 conc in semi-log steps)

Cpd Submission

100 x Stock solution in 100% DMSO or
pre-weighed powder (request guidelines)

Report

Detailed report for each project
Sample report will be provided upon request

Turnaround Time

No fixed time slots; first come - first served;
routinely within 10 working days

Info Sheets

Method: Radiometric Assay, Method: ATP-Glo™ Assay

List of Kinases for this Service

PDF

Guidelines for Cpd Submission

Guidelines       SPF       CSF

Free Choice Kinase Assay Projects / Kinase Assays | ProQinase – Drug Discovery in Oncology

Error

The website encountered an unexpected error. Please try again later.