Biochemical Assay Services

Free Choice Kinase Assay Projects / Kinase Assays

Field of Application

Free choice kinase assay projects allow characterization of your test compounds in a total flexible mode. For each project you can freely define (i) the number of kinase assays, (ii) the number of test compounds (iii) and the number of data points for each test compound (i.e. number of concentrations and replicates). All kinase assays are designed to measure biochemical kinase activity.

Our Products

Number Kinase Synonyms
1 ABL1 E255K ABL1, c-Abl, JTK7, p150
2 ABL1 F317I ABL1, ABL, JTK7, p150, c-ABL, v-abl
3 ABL1 G250E ABL1, ABL, JTK7, p150, c-ABL, v-abl
4 ABL1 H396P ABL1, ABL, JTK7, p150, c-ABL, v-abl
5 ABL1 M351T ABL1, ABL, JTK7, p150, c-ABL, v-abl
6 ABL1 Q252H ABL1, ABL, JTK7, p150, c-ABL, v-abl
7 ABL1 T315I ABL1, ABL, JTK7, p150, c-ABL, v-abl
8 ABL1 wt ABL1, ABL, JTK7, p150, c-ABL, v-abl
9 ABL1 Y253F ABL1, ABL, JTK7, p150, c-ABL, v-abl
10 ABL2 ABL2, ABLL, ARG
11 ACK1 TNK2, ACK, p21cdc42Hs, Activated CDC42 kinase 1
12 ACV-R1 ACVR1, ACTRI, ACVRLK2, ALK2, SKR1
13 ACV-R1B ACVR1B, ACTRIB, ACVRLK4, ALK4, SKR2
14 ACV-R2A ACVR2, ACTRII
15 ACV-R2B ActR-IIB, ACTRIIB
16 ACV-RL1 ACVRL1, ACVRLK1, ALK-1, ALK1, HHT, HHT2, ORW2, SKR3
17 AKT1 aa1-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
18 AKT1 aa106-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
19 AKT2 aa1-481 AKT2, PKBB, PKBBETA, PKB beta, PRKBB, RAC-beta, RAC-PK-beta
20 AKT2 aa107-481 AKT2, PRKBB, PKBBETA, RAC-BETA
21 AKT3 aa1-479 AKT3, PKBG, PKB gamma, PRKBG, RAC-gamma, RAC-PK-gamma, STK-2, DKFZp434N0250
22 AKT3 aa106-479 AKT3, PKBG, PRKBG, STK-2, RAC-gamma, RAC-PK-gamma
23 ALK C1156Y (GST-HIS-tag) ALK, CD246, NBLST3
24 ALK F1174L (GST-HIS-tag) ALK, CD246, NBLST3
25 ALK F1174S (GST-HIS-tag) ALK, CD246, NBLST3
26 ALK G1202R (GST-HIS-tag) ALK, CD246, NBLST3
27 ALK L1196M (GST-HIS-tag) ALK, CD246, NBLST3
28 ALK R1275Q (GST-HIS-tag) ALK, CD246, NBLST3
29 ALK wt (GST-HIS-tag) ALK, CD246, NBLST3
30 AMPK-alpha1 aa1-550 PRKAA1, MGC33776, MGC57364
31 ARK5 NUAK1, KIAA0537
32 ASK1 MAP3K5, ASK1, MAPKKK5, MEKK5
33 Aurora-A AURKA, AIK, ARK1, AURA, BTAK, STK15, MGC34538, STK6
34 Aurora-B AURKB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AIM-1, STK12
35 Aurora-C AURKC, AIE2, AIK3, STK13
36 AXL AXL, EC, UFO
37 B-RAF V600E BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
38 B-RAF wt BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
39 BLK BLK, n/a
40 BMPR1B BMPR1B, ALK6, CDw293
41 BMX BMX, ETK, PSCTK2, PSCTK3
42 BRK PTK6, n/a
43 BRSK1 BRSK1, KIAA1811
44 BRSK2 C11orf7, FLJ41362, HUSSY-12, PEN11B, SAD1, STK29
45 BTK BTK, AGMX1, AT, ATK, BPK, PSCTK1
46 BUB1B BUB1B, BUBR1, Bub1A, MAD3L, hBUBR1
47 CAMK1D CAMK1D, CKLiK, CaM-K1, CaMKID
48 CAMK2A CAMK2A, CAMKA, KIAA0968
49 CAMK2B CAMK2B, CAM2, CAMK2, CAMKB, MGC29528
50 CAMK2D CAMK2D, CAMKD, MGC44911, CaMKII delta
51 CAMK2G CAMK2G, CAMK, CAMK-II, CAMKG, MGC26678
52 CAMK4 CAMK4, CaMK-GR, MGC36771
53 CAMKK1 CAMKK1, CAMKKA, DKFZp761M0423, MGC34095
54 CAMKK2 CAMKK2, CAMKK, CAMKKB, KIAA0787, MGC15254
55 CCDC6-RET CCDC6-RET, CCDC6-RETa
56 CDC42BPA CDC42BPA, MRCK-alpha
57 CDC42BPB CDC42BPB, MRCK-beta, MRCKb
58 CDC7/DBF4 CDC7, CDC7L1, HsCdc7, HsCDC7, Hsk1, huCdc7
59 CDK1/CycA2 CDC2, p34
60 CDK1/CycB1 CDC2, p34
61 CDK1/CycE1 CDC2, p34
62 CDK12 R722C/CycK CDK12, CRKRS, CRK7
63 CDK12 wt/CycK CDK12, CRKRS, CRK7
64 CDK13/CycK CDK13, CDC2L, CDC2L5, CHED
65 CDK16/CycY CDK16, PCTAIRE1, PCTAIRE, PCTGAIRE, PCTK1
66 CDK17/p35NCK CDK17, PCTAIRE2, PCTK2
67 CDK18/CycY CDK18, PCTAIRE, PCTAIRE3, PCTK3
68 CDK19/CycC CDK19, CDC2L6, CDK11
69 CDK2/CycA2 CDK2, p33(CDK2)
70 CDK2/CycD1 CDK2, p33
71 CDK2/CycE1 CDK2, p33(CDK2)
72 CDK20/CycH CDK20, CAK-kinase p42
73 CDK20/CycT1 CDK20, CAK-kinase p42, CCRK, CDCH, p42, PNQALRE
74 CDK3/CycC CDK3, CDKN3
75 CDK3/CycE1 CDK3, n/a
76 CDK4/CycD1 CDK4, CMM3, PSK-J3, MGC14458
77 CDK4/CycD2 CDK4, CMM3, PSK-J3
78 CDK4/CycD3 CDK4, CMM3, PSK-J3, MGC14458
79 CDK5/p25NCK CDK5, PSSALRE
80 CDK5/p35NCK CDK5, PSSALRE
81 CDK6/CycD1 CDK6, PLSTIRE, MGC59692
82 CDK6/CycD2 CDK6, PLSTIRE
83 CDK6/CycD3 CDK6, PLSTIRE
84 CDK7/CycH/MAT1 CDK7, CAK1, CDKN7, STK1, p39MO15
85 CDK8/CycC CDK8, K35
86 CDK9/CycK CDK9, C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase
87 CDK9/CycT1 CDK9, C-2k, CDC2L4K35, PITALRE, TAK
88 CHK1 CHEK1, n/a
89 CHK2 CHEK2, CDS1, HuCds1, PP1425, RAD53, bA444G7
90 CK1-alpha1 CSNK1A1, CK1, HLCDGP1, PRO2975
91 CK1-delta CSNK1D, HCKID
92 CK1-epsilon CSNK1E, CKIe, HCKIE, MGC10398
93 CK1-gamma1 CSNK1G1
94 CK1-gamma2 CSNK1G2, CK1g2
95 CK1-gamma3 CSNK1G3
96 CK2-alpha1 CSNK2A1, CKII, CK2A1
97 CK2-alpha2 CSNK2A2, n/a
98 CLK1 CLK1, CLK, CLK/STY
99 CLK2 CLK2, MGC61500, clk2, hCLK2
100 CLK3 CLK3, PHCLK3, PHCLK3/152
101 CLK4 CLK4, DKFZp686A20267, CDC-like kinase 4
102 COT MAP3K8, EST, ESTF, TPL2, Tpl-2, c-COT
103 CSF1-R CSF1R, C-FMS, CD115, CSF-1-R, CSFR, FIM2, FMS
104 CSK CSK, n/a
105 DAPK1 DAPK1, n/a
106 DAPK2 DAPK2, DRP-1
107 DAPK3 DAPK3, ZIP, ZIPK
108 DCAMKL2 DCLK2, DCLK, KIAA0369
109 DDR2 N456S DDR2, MIG20a, NTRKR3, TKT, TYRO10
110 DDR2 T654M DDR2, MIG20a, NTRKR3, TKT, TYRO10
111 DDR2 wt DDR2, MIG20a, NTRKR3, TKT, TYRO10
112 DMPK DMPK, DM, DM1, DM1PK, DMK
113 DNA-PK PRKDC, DNAPK, DNPK1, HYRC, HYRC1, XRCC7, p350
114 DYRK1A DYRK1A, DYRK, DYRK1, HP86, MNB, MNBH
115 DYRK1B DYRK1B, MIRK
116 DYRK2 DYRK2
117 DYRK3 DYRK3, DYRK5, RED, REDK
118 DYRK4 DYRK4
119 EEF2K EEF2K, HSU93850, MGC45041, eEF-2K
120 EGF-R C797S EGF-R, ERBB, ERBB1
121 EGF-R d746-750 EGFR, ERBB, mENA, ERBB1
122 EGF-R d747-749/A750P EGFR, ERBB, mENA, ERBB1
123 EGF-R d747-752/P753S EGFR, ERBB, mENA, ERBB1
124 EGF-R d752-759 EGFR, ERBB, mENA, ERBB1
125 EGF-R G719C EGFR, ERBB, mENA, ERBB1
126 EGF-R G719S EGFR, ERBB, mENA, ERBB1
127 EGF-R L858R EGFR, ERBB, ERBB1
128 EGF-R L861Q EGFR, ERBB, mENA, ERBB1
129 EGF-R T790M EGFR, ERBB, ERBB1
130 EGF-R T790M/L858R EGFR, ERBB, ERBB1
131 EGF-R wt EGFR, ERBB, mENA, ERBB1
132 EIF2AK2 EIF2AK2, EIF2AK1, PKR, PRKR
133 EIF2AK3 EIF2AK3, DKFZp781H1925, PEK, PERK, WRS
134 EML4 ALK ALK
135 EML4 ALK F1174L ALK
136 EPHA1 EPHA1, EPH, EPHT, EPHT1
137 EPHA2 EPHA2, ECK
138 EPHA3 EPHA3, ETK, ETK1, EphA3, HEKECK, HEK4, TYRO4
139 EPHA4 EPHA4, HEK8, SEK, TYRO1
140 EPHA5 EPHA5, CEK7, EHK1, EphA5, HEK7, Hek7, TYRO4
141 EPHA6 EPHA6, EHK2, EHK-2, EPA6
142 EPHA7 EPHA7, EHK3, HEK11
143 EPHA8 EPHA8, EEK, EphA8, HEK3, KIAA1459
144 EPHB1 EPHB1, ELK, NET, Hek6, EPHT2
145 EPHB2 EPHB2, DRT, ERK, Hek5, EPHT3, Tyro5
146 EPHB3 EPHB3, ETK2, HEK2, TYRO6
147 EPHB4 EPHB4, HTK, MYK1, TYRO11
148 ERBB2 775YVMA776 ERBB2, CD340, HER2, MLN19, NGL, TKR1
149 ERBB2 wt ERBB2, NEU, NGL, HER2, TKR1, HER-2
150 ERBB4 ERBB4, n/a
151 ERK1 MAPK3, ERT2, HS44KDAP, HUMKER1A, P44ERK1, P44MAPK, PRKM3
152 ERK2 MAPK1, ERK, ERT1, MAPK2, P42MAPK, PRKM1, PRKM2, p38, p40, p41
153 ERK5 MAPK7, BMK1, ERK4, PRKM7
154 ERK7 MAPK15, ERK8, MAPK15
155 FAK aa2-1052 PTK2, FADK, pp125FAK
156 FER FER, TYK3, c-FER, p94-FER
157 FES FES, FPS
158 FGF-R1 V561M FGFR1, FGFR-1, bFGF-R, FLT2, CEK, CD331
159 FGF-R1 wt FGFR1, H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM
160 FGF-R2 FGFR2, FGFR2, BEK, BFR-1, CD332, CEK3, CFD1, ECT1, FGFR-2, JWS, KGFR, KSAM, K-SAM, TK14, TK25
161 FGF-R3 G697C FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
162 FGF-R3 K650E FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
163 FGF-R3 K650M FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
164 FGF-R3 wt FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
165 FGF-R4 FGFR4, TKF, JTK2, MGC20292
166 FGR FGR, SRC2, c-fgr, p55c-fgr
167 FLT3 D835Y FLT3, CD135, FLK2, STK-1, STK1
168 FLT3 ITD FLT3, CD135, FLK2, STK-1, STK1
169 FLT3 wt FLT3, CD135, FLK2, STK-1, STK1
170 FRK FRK, GTK, PTK5, RAK
171 FYN wt FYN, SLK, SYN, p59-Fyn
172 FYN Y531F FYN, SLK, SYN, p59-FYN, cFYN
173 GRK2 ADRBK1
174 GRK3 ADRBK2
175 GRK4 GRK4, GPRK2L, GPRK4, GRK4a, IT11
176 GRK5 GRK5
177 GRK6 GRK6
178 GRK7 GRK7
179 GSG2 GSG2, Haspin
180 GSK3-alpha GSK3A
181 GSK3-beta GSK3B
182 HCK HCK, JTK9
183 HIPK1 HIPK1, KIAA0630, MGC26642, MGC33446, MGC33548, Myak, Nbak2
184 HIPK2 HIPK2, PRO0593
185 HIPK3 HIPK3, ANPK, DYRK6, FIST, FIST3, PKY, YAK1
186 HIPK4 HIPK4, FLJ32818
187 HRI EIF2AK1, HCR
188 IGF1-R IGF1R, JTK13
189 IKK-alpha CHUK, IKBKA, IKK1, IKKA, NFKBIKA, TCF16
190 IKK-beta IKBKB, IKK2, IKKB, NFKBIKB
191 IKK-epsilon IKBKE, IKKE, IKKI, IKK-i, KIAA0151
192 INS-R INSR, n/a
193 INSR-R INSRR, IRR
194 IRAK1 IRAK1, IRAK, Pelle
195 IRAK4 (untagged) IRAK4, REN64, NY-REN-64
196 ITK ITK, EMT 2, LYK 2, PSCTK2 2, IL2-inducible T-cell kinase
197 JAK1 aa583-1154 S729C JAK1, JAK1A, JAK1B, JTK3
198 JAK1 aa583-1154 wt JAK1, JAK1A, JAK1B, JTK3
199 JAK2 JAK2, n/a
200 JAK3 JAK3, JAKL, L-JAK, LJAK
201 JNK1 MAPK8, PRKM8, SAPK1, JNK1-alpha1
202 JNK2 MAPK9, PRKM9, p54aSAPK, JNK2-alpha2
203 JNK3 MAPK10, JNK3A, p54bSAPK
204 KIT A829P KIT, C-Kit, PBT, CD117, SCFR, c-kit
205 KIT D816H KIT, C-Kit, PBT, CD117, SCFR, c-kit
206 KIT D816V KIT, C-Kit, PBT, CD117, SCFR, c-kit
207 KIT T670I KIT, CD117, SCFR, PBT, C-Kit
208 KIT V559D KIT, C-Kit, PBT, CD117, SCFR, c-kit
209 KIT V559D/T670I KIT, C-Kit, PBT, CD117, SCFR, c-kit
210 KIT V559D/V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
211 KIT V560G KIT, C-Kit, PBT, CD117, SCFR, c-kit
212 KIT V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
213 KIT wt KIT, C-Kit, PBT, CD117, SCFR, c-kit
214 LCK LCK, n/a
215 LIMK1 LIMK1, LIMK
216 LIMK2 LIMK2
217 LRRK2 G2019S LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
218 LRRK2 I2020T LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
219 LRRK2 R1441C LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
220 LRRK2 wt LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
221 LTK LTK, TYK1
222 LYN LYN, JTK8
223 MAP3K1 MAP3K1, MAPKKK1, MEKK, MEKK1
224 MAP3K10 MAP3K10, MLK2, MST, MEKK10
225 MAP3K11 MAP3K11, MGC17114, MLK-3, PTK1, SPRK
226 MAP3K7/MAP3K7IP1 MAP3K7, TAK1, TGF1a, MEKK7
227 MAP3K9 MAP3K9, MLK1, PRKE1, MEKK9
228 MAP4K2 MAP4K2, BL44, GCK, RAB8IP
229 MAP4K4 MAP4K4, HGK, MEKKK4, NIK
230 MAP4K5 MAP4K5, KHS1, GCKR, KHS, MAPKKKK5
231 MAPKAPK2 MAPKAPK2, n/a
232 MAPKAPK3 MAPKAPK3, 3PK, MAPKAP, MAPKAP3
233 MAPKAPK5 MAPKAPK5, PRAK
234 MARK1 MARK1, KIAA1477
235 MARK2 MARK2, EMK1, MGC99619, PAR-1, ELKL motif kinase 1
236 MARK3 MARK3, CTAK1, KP78, PAR1A
237 MARK4 MARK4, KIAA1860, MARKL1
238 MASTL MASTL, GLW, GREATWALL, GWL, hGWL, MAST-L, THC2
239 MATK MATK, CHK, CTK, DKFZp434N1212, HHYLTK, HYL, Lsk, MGC1708, MGC2101
240 MEK1 F53L MAP2K1, MAP2K1, MAPKK1, MAPKK 1, MKK1, PRKMK1
241 MEK1 wt MAP2K1, MAPKK1, MKK1, PRKMK1
242 MEK2 MAP2K2, MAPKK2, MKK2, PRKMK2
243 MEK5 MAP2K5, MAP2K5, MAPKK5, MKK5, PRKMK5
244 MEKK2 MAP3K2, MAPKKK2, MEKK2B
245 MEKK3 MAP3K3, MAPKKK3, MEK kinase3
246 MELK MELK, PK38
247 MERTK MERTK, MER, MER-PEN, RP38
248 MET D1228H MET, HGFR, RCCP2
249 MET D1228N MET, HGFR, RCCP2
250 MET F1200I MET, HGFR, RCCP2
251 MET G1163R MET, HGFR, RCCP2
252 MET L1195V MET, HGFR, RCCP2
253 MET M1250T MET, HGFR, RCCP2
254 MET wt MET, HGFR, RCCP2
255 MET Y1230A MET, HGFR, RCCP2
256 MET Y1230C MET, HGFR, RCCP2
257 MET Y1230D MET, HGFR, RCCP2
258 MET Y1230H MET, HGFR, RCCP2
259 MET Y1235D MET, HGFR, RCCP2
260 MINK1 MINK1, B55, YSK2, MAP4K6, ZC3
261 MKK4 MAP2K4, JNKK, JNKK1, MAPKK4, MEK4, PRKMK4, SEK, SERK1
262 MKK6 S207D/T211D MAP2K6, MAPKK6, MEK6, MKK6, PRKMK6, SAPKK3
263 MKK7 MAP2K7, MAPKK7, MEK7, PRKMK7
264 MKNK1 MKNK1, MNK1
265 MKNK2 MKNK2, MNK2, GPRK7
266 MLK4 n/a, KIAA1804
267 MST1 STK4, KRS2, YSK3
268 MST2 STK3, MST-2, KRS1
269 MST3 STK24, MST-3, MST3B, STK3
270 MST4 MST4, MASK
271 mTOR FRAP1, FRAP, FRAP2, RAFT1, RAPT1, rapamycin target protein
272 MUSK MUSK, n/a
273 MYLK MYLK, smMLCK, FLJ12216, KRP, MLCK, MLCK108, MLCK210
274 MYLK2 MYLK2, KMLC, MLCK, skMLCK
275 MYLK3 MYLK3, caMLCK, MLCK2, MYLK2
276 NEK1 NEK1, NY-REN-55
277 NEK11 NEK11, FLJ23495
278 NEK2 NEK2, NLK1, HsPK21, HsPK 21
279 NEK3 NEK3, HSPK36, MGC29949
280 NEK4 NEK4, NRK2, STK2
281 NEK6 NEK6, SID6-1512
282 NEK7 NEK7, n/a
283 NEK9 NEK9, DKFZp434D0935, MGC16714, NERCC, NERCC1, Nek8
284 NIK MAP3K14, FTDCR1B, HS, HSNIK
285 NLK NLK, n/a
286 NPM1 ALK n/a, n/a
287 NPM1 ALK F1174L n/a, n/a
288 p38-alpha MAPK14, p38-alpha
289 p38-beta MAPK11, p38-beta
290 p38-delta MAPK13, n/a
291 p38-gamma MAPK12, ERK-6, ERK3, ERK5, ERK6, PRKM12, SAPK-3, SAPK3
292 PAK1 PAK1, PAKalpha
293 PAK2 PAK2, PAK65, PAKgamma
294 PAK3 PAK3, CDKN1A, MRX30, OPHN3, PAK3beta, bPAK, hPAK3
295 PAK4 PAK4, n/a
296 PAK6 PAK6, PAK5
297 PAK7 PAK7, KIAA1264, MGC26232
298 PASK PASK, DKFZP434O051, DKFZp686P2031, KIAA0135, PASKIN, STK3
299 PBK PBK, TOPK, SPK, Nori-3, FLJ14385
300 PDGFR-alpha D842V PDGFRA, PDGFR2, CD140a
301 PDGFR-alpha T674I PDGFRA, PDGFR2, CD140a
302 PDGFR-alpha V561D PDGFRA, PDGFR2, CD140a
303 PDGFR-alpha wt PDGFRA, PDGFR2, CD140a
304 PDGFR-beta PDGFRB, JTK12, PDGFR, CD140B, PDGFR1, PDGF-R-beta
305 PDK1 PDPK1, PKB-like
306 PHKG1 PHKG1, PHKg1
307 PHKG2 PHKG2, PHKg2
308 PI4K2A PI4K2A, PI4KII, PIK42A, RP11-548K23.6
309 PI4K2B PI4K2B, PI4KIIB, PI4KII-BETA, PIK42B
310 PI4KB PI4KB, NPIK, pi4K92, PI4K92, PI4Kbeta, PI4KBETA, PI4K-beta, PI4K-BETA, PI4KIIIBETA, PIK4CB
311 PIK3C2A PIK3C2A, CPK, MGC142218, PI3-K-C2A
312 PIK3C2B PIK3C2B, C2-PI3K, PI3K-C2beta
313 PIK3C2G PIK3C2G, PI3K-C2GAMMA, PI3K-C2-gamma
314 PIK3C3 PIK3C3, hVps34, MGC61518, PI3-kinase type 3, PI3K type 3, Vps34, VPS34
315 PIK3CA/PIK3R1 PIK3CA, MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha
316 PIK3CB D1067A/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
317 PIK3CB D1067V/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
318 PIK3CB D1067Y/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
319 PIK3CB E1051K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
320 PIK3CB E633K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
321 PIK3CB L1049R/PIK3R1 PIK3CB
322 PIK3CB wt/PIK3R1 PIK3CB, PI3K, PI3KBETA, PI3K-beta, PIK3C1, p110-beta
323 PIK3CD/PIK3R1 PIK3CD, p110D, P110DELTA, PI3K, PI3K-delta, p110-delta
324 PIK3CG PIK3CG, p120-PI3K, PI3CG, PI3K, PI3Kgamma, PI3K-gamma, p110-gamma
325 PIM1 PIM1, PIM
326 PIM2 PIM2, n/a
327 PIM3 PIM3, n/a
328 PIP5K1A PIP5K1A, PIP5K1-alpha, PIP5KIalpha, PtdIns(4)P-5-kinase 1 alpha
329 PIP5K1B PIP5K1B, MSS4, PIP5K1-beta, STM7
330 PIP5K1C PIP5K1C, PIP5K1-gamma, PIP5Kgamma, PIP5K-GAMMA, PIPKIg_v4
331 PKA PRKACA, MGC48865, PKA
332 PKC-alpha PRKCA, PKCA, PRKACA, PKC-alpha
333 PKC-beta1 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
334 PKC-beta2 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
335 PKC-delta PRKCD, MAY1, MGC49908, nPKC-delta
336 PKC-epsilon PRKCE, PKCE, nPKC-epsilon
337 PKC-eta PRKCH, PKC-L, PKCL, PRKCL, nPKC-eta
338 PKC-gamma PRKCG, PKCC, PKCG, SCA14, MGC57564
339 PKC-iota PRKCI, PKCI, DXS1179E, MGC26534, nPKC-iota
340 PKC-mu PRKD1, PKD, PKCM, PKC-MU
341 PKC-nu PRKD3, EPK2
342 PKC-theta PRKCQ, PRKCT, nPKC-theta
343 PKC-zeta PRKCZ, PKC2
344 PKC-zeta wt aa184-592 (PKM-zeta) PRKCZ, PKM-zeta, nPKC-zeta, PKC2
345 PKMYT1 PKMYT1, MYT1
346 PKN3 PKN3, PKNbeta, RP11-545E17.1
347 PLK1 PLK1, PLK, STPK13
348 PLK3 PLK3, CNK, FNK, PRK
349 PRK1 PKN1, DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204
350 PRK2 PKN2, PRKCL2, PAK-2
351 PRKD2 PRKD2, PKD2, HSPC187
352 PRKG1 PRKG1, PKG1, CGKI, MGC71944, PGK, PRKG1B, PRKGR1B, cGKIBETA, cGKI-alph
353 PRKG2 PRKG2, PKG2, PRKGR2, cGKII
354 PRKX PRKX, PKX1
355 PYK2 PTK2B, CADTK, CAKB, FADK2, FAK2, PKB, PTK, PYK2, RAFTK, CAK beta
356 RAF1 Y340D/Y341D (untagged) RAF1, c-RAF
357 RET E762Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
358 RET G691S RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
359 RET M918T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
360 RET R749T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
361 RET R813Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
362 RET S891A RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
363 RET V804E RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
364 RET V804L RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
365 RET V804M RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
366 RET wt RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
367 RET Y791F RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
368 RET Y806H RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
369 RIPK2 RIPK2, CARD3, CARDIAK, CCK, GIG30, RICK, RIP-2, RIP2
370 RIPK4 RIPK4, ANKK2, ANKRD3, DIK, MGC129992, MGC129993, PKK, RIP4
371 RIPK5 DSTYK, SgK496, SHIK
372 ROCK1 ROCK1, P160ROCK
373 ROCK2 ROCK2, KIAA0619, ROC2
374 RON MST1R, CD136, CDw136, PTK8
375 ROS ROS1, MCF3
376 RPS6KA1 RPS6KA1, RSK3, HU-1, MAPKAPK1A, RSK, RSK1
377 RPS6KA2 RPS6KA2, RSK1, HU-2, MAPKAPK1C, RSK, RSK3
378 RPS6KA3 RPS6KA3, HU-2, HU-3, ISPK-1, MAPKAPK1B, MRX19, RSK, RSK2
379 RPS6KA4 RPS6KA4, MSK2, RSK-B
380 RPS6KA5 RPS6KA5, MSK1, EC 2.7.11, MGC1911, MSPK1, RLPK, RSKL
381 RPS6KA6 RPS6KA6, RSK4
382 S6K RPS6KB1, S6K1, STK14A
383 S6K-beta RPS6KB2, KLS, P70-beta-1, P70-beta-2, S6K-beta2, S6K2, SRK, p70S6Kb
384 SAK PLK4, SAK, STK18
385 SGK1 SGK, n/a
386 SGK2 SGK2, H-SGK2, dJ138B7.2
387 SGK3 SGKL, CISK, SGK2, SGK3
388 SIK1 SIK1, MSK, SNF1LK, SIK, SIK-1, SNF1LK
389 SIK2 SIK2, QIK, SNF1LK2
390 SIK3 SIK3, L19, QSK, SIK-3
391 SLK SLK, KIAA0204, STK2, bA16H23.1, se20-9
392 SNARK NUAK2, DKFZp434J037
393 SNK PLK2, SNK
394 SRC (GST-HIS-tag) SRC, ASV, SRC1, c-SRC, p60-Src
395 SRMS SRMS, C20orf148, SRM, dJ697K14.1
396 SRPK1 SRPK1, SFRSK1
397 SRPK2 SRPK2, SFRSK2
398 STK17A STK17A, DRAK1
399 STK23 SRPK3, MSSK1, MGC102944
400 STK25 STK25, DKFZp686J1430, SOK1, YSK1
401 STK33 STK33
402 STK39 STK39, STLK3, DCHT, SPAK
403 SYK aa1-635 SYK, n/a
404 TAOK2 TAOK2, KIAA0881, MAP3K17, PSK, PSK1, TAO1, TAO2
405 TAOK3 TAOK3, DPK, JIK, MAP3K18, TAO kinase 3
406 TBK1 TBK1, CDC37, HSPCA, HSPCB, IKBKG, NAK, T2K, TANK, TRAF2
407 TEC TEC, PSCTK4
408 TGFB-R1 TGFBR1, ALK5, ACVRLK4
409 TGFB-R2 TGFBR2, HNPCC6, MFS2, RIIC, TGFR-2, TGFbeta-RII
410 TIE2 R849W TEK, VMCM, TIE-2, VMCM1, CD202B
411 TIE2 wt TEK, VMCM, TIE-2, VMCM1, CD202B
412 TIE2 Y1108F TEK, VMCM, TIE-2, VMCM1, CD202B
413 TIE2 Y897S TEK, VMCM, TIE-2, VMCM1, CD202B
414 TLK1 TLK1, PKU-beta, KIAA0137
415 TLK2 TLK2, MGC44450, PKU-ALPHA
416 TNK1 TNK1, n/a
417 TRK-A G667C MTC, TRK1, TRKA
418 TRK-A wt NTRK1, MTC, TRK, TRK1, TRKA
419 TRK-B NTRK2, GP145-TrkB, TRKB, Trk-B
420 TRK-C NTRK3, GP145-TrkC, TRKC, Trk-C
421 TSF1 STK16, KRCT, MPSK, PKL12
422 TSK2 TSSK2, DGS-G, SPOGA2, FLJ38613
423 TSSK1 TSSK1, FKSG81, SPOGA4, STK22D
424 TTBK1 aa1-1321 TTBK1, BDTK
425 TTBK1 aa1-480 TTBK1, BDTK
426 TTBK2 TTBK2, BDTK, KIAA1855, RP3-330M21.4
427 TTK TTK, ESK, MPS1L1, PYT
428 TXK TXK, BTKL, PSCTK5, PTK4, RLK
429 TYK2 TYK2, JTK1
430 TYRO3 TYRO3, BYK, Brt, Dtk, Sky, Tif
431 ULK2 ULK2, ATG1B, KIAA0623, Unc51.2
432 VEGF-R1 FLT1, FLT, VEGFR1
433 VEGF-R2 KDR, FLK1, VEGFR, VEGFR2
434 VEGF-R3 FLT4, PCL, VEGFR3
435 VRK1 VRK1, n/a
436 VRK2 VRK2, n/a
437 WEE1 WEE1, WEE1hu
438 WNK1 WNK1, KDP, KIAA0344, PHA2C, PRKWNK1
439 WNK2 WNK2, KIAA1760, NY-CO-43, P/OKcl.13, PRKWNK2, SDCCAG43
440 WNK3 WNK3, KIAA1566, PRKWNK3
441 YES YES, C-YES, HsT441, P61-YES
442 ZAK MLTK, mlklak, AZK
443 ZAP70 ZAP70, SRK, STD, TZK, ZAP-70

Info in Brief

Kinase Panel

444 kinases, including 91 disease-relevant kinase
mutants and 20 lipid kinases

Assay Technologies

Protein kinases: FlashPlate™-based radiometric assay;
lipid kinases: ADP-Glo™ assay technology (Promega)

ATP conc

App. ATP-Km for each kinase

Testing Modes

Single concentration measurement or IC50 profiling
(10 conc in semi-log steps)

Cpd Submission

100 x Stock solution in 100% DMSO or
pre-weighed powder (request guidelines)

Report

Detailed report for each project
Sample report will be provided upon request

Turnaround Time

No fixed time slots; first come - first served;
routinely within 10 working days

Info Sheets

Method: Radiometric Assay, Method: ATP-Glo™ Assay

List of Kinases for this Service

PDF

Guidelines for Cpd Submission

Guidelines       SPF       CSF