Biochemical Assay Services

Free Choice Kinase Assay Projects

Field of Application

Free choice kinase assay projects allow characterization of your test com-pounds in a self-selected panel of biochemical kinase activity assays. For each project you can freely define (i) the number of test compounds, (ii) the kinase panel, (iii) and the number of data points for each test compound (i.e. number of concentrations and replicates).

Our Products

Number Kinase Synonyms
1 ABL1 E255K ABL1, c-Abl, JTK7, p150
2 ABL1 F317I ABL1, ABL, JTK7, p150, c-ABL, v-abl
3 ABL1 G250E ABL1, ABL, JTK7, p150, c-ABL, v-abl
4 ABL1 H396P ABL1, ABL, JTK7, p150, c-ABL, v-abl
5 ABL1 M351T ABL1, ABL, JTK7, p150, c-ABL, v-abl
6 ABL1 Q252H ABL1, ABL, JTK7, p150, c-ABL, v-abl
7 ABL1 T315I ABL1, ABL, JTK7, p150, c-ABL, v-abl
8 ABL1 wt ABL1, ABL, JTK7, p150, c-ABL, v-abl
9 ABL1 Y253F ABL1, ABL, JTK7, p150, c-ABL, v-abl
10 ABL2 ABL2, ABLL, ARG
11 ACK1 TNK2, ACK, p21cdc42Hs, Activated CDC42 kinase 1
12 ACV-R1 ACVR1, ACTRI, ACVRLK2, ALK2, SKR1
13 ACV-R1B ACVR1B, ACTRIB, ACVRLK4, ALK4, SKR2
14 ACV-R2A ACVR2, ACTRII
15 ACV-R2B ActR-IIB, ACTRIIB
16 ACV-RL1 ACVRL1, ACVRLK1, ALK-1, ALK1, HHT, HHT2, ORW2, SKR3
17 AKT1 aa1-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
18 AKT1 aa106-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
19 AKT2 aa1-481 AKT2, PKBB, PKBBETA, PKB beta, PRKBB, RAC-beta, RAC-PK-beta
20 AKT2 aa107-481 AKT2, PRKBB, PKBBETA, RAC-BETA
21 AKT3 aa1-479 AKT3, PKBG, PKB gamma, PRKBG, RAC-gamma, RAC-PK-gamma, STK-2, DKFZp434N0250
22 AKT3 aa106-479 AKT3, PKBG, PRKBG, STK-2, RAC-gamma, RAC-PK-gamma
23 ALK C1156Y (GST-HIS-tag) ALK, CD246, NBLST3
24 ALK F1174L (GST-HIS-tag) ALK, CD246, NBLST3
25 ALK F1174S (GST-HIS-tag) ALK, CD246, NBLST3
26 ALK G1202R (GST-HIS-tag) ALK, CD246, NBLST3
27 ALK L1196M (GST-HIS-tag) ALK, CD246, NBLST3
28 ALK R1275Q (GST-HIS-tag) ALK, CD246, NBLST3
29 ALK wt (GST-HIS-tag) ALK, CD246, NBLST3
30 AMPK-alpha1 aa1-550 PRKAA1, MGC33776, MGC57364
31 ARK5 NUAK1, KIAA0537
32 ASK1 MAP3K5, ASK1, MAPKKK5, MEKK5
33 Aurora-A AURKA, AIK, ARK1, AURA, BTAK, STK15, MGC34538, STK6
34 Aurora-B AURKB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AIM-1, STK12
35 Aurora-C AURKC, AIE2, AIK3, STK13
36 AXL AXL, EC, UFO
37 B-RAF V600E BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
38 B-RAF wt BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
39 BLK BLK, n/a
40 BMPR1A BMPR1A, ACVRLK3, ALK3
41 BMPR1B BMPR1B, ALK6, CDw293
42 BMX BMX, ETK, PSCTK2, PSCTK3
43 BRK PTK6, n/a
44 BRSK1 BRSK1, KIAA1811
45 BRSK2 C11orf7, FLJ41362, HUSSY-12, PEN11B, SAD1, STK29
46 BTK BTK, AGMX1, AT, ATK, BPK, PSCTK1
47 BUB1B BUB1B, BUBR1, Bub1A, MAD3L, hBUBR1
48 CAMK1D CAMK1D, CKLiK, CaM-K1, CaMKID
49 CAMK2A CAMK2A, CAMKA, KIAA0968
50 CAMK2B CAMK2B, CAM2, CAMK2, CAMKB, MGC29528
51 CAMK2D CAMK2D, CAMKD, MGC44911, CaMKII delta
52 CAMK2G CAMK2G, CAMK, CAMK-II, CAMKG, MGC26678
53 CAMK4 CAMK4, CaMK-GR, MGC36771
54 CAMKK1 CAMKK1, CAMKKA, DKFZp761M0423, MGC34095
55 CAMKK2 CAMKK2, CAMKK, CAMKKB, KIAA0787, MGC15254
56 CCDC6-RET CCDC6-RET, CCDC6-RETa
57 CDC42BPA CDC42BPA, MRCK-alpha
58 CDC42BPB CDC42BPB, MRCK-beta, MRCKb
59 CDC7/DBF4 CDC7, CDC7L1, HsCdc7, HsCDC7, Hsk1, huCdc7
60 CDK1/CycA2 CDC2, p34
61 CDK1/CycB1 CDC2, p34
62 CDK1/CycE1 CDC2, p34
63 CDK12 R722C/CycK CDK12, CRKRS, CRK7
64 CDK12 wt/CycK CDK12, CRKRS, CRK7
65 CDK13/CycK CDK13, CDC2L, CDC2L5, CHED
66 CDK16/CycY CDK16, PCTAIRE1, PCTAIRE, PCTGAIRE, PCTK1
67 CDK17/p35NCK CDK17, PCTAIRE2, PCTK2
68 CDK18/CycY CDK18, PCTAIRE, PCTAIRE3, PCTK3
69 CDK19/CycC CDK19, CDC2L6, CDK11
70 CDK2/CycA2 CDK2, p33(CDK2)
71 CDK2/CycD1 CDK2, p33
72 CDK2/CycE1 CDK2, p33(CDK2)
73 CDK20/CycH CDK20, CAK-kinase p42
74 CDK20/CycT1 CDK20, CAK-kinase p42, CCRK, CDCH, p42, PNQALRE
75 CDK3/CycC CDK3, CDKN3
76 CDK3/CycE1 CDK3, n/a
77 CDK4/CycD1 CDK4, CMM3, PSK-J3, MGC14458
78 CDK4/CycD2 CDK4, CMM3, PSK-J3
79 CDK4/CycD3 CDK4, CMM3, PSK-J3, MGC14458
80 CDK5/p25NCK CDK5, PSSALRE
81 CDK5/p35NCK CDK5, PSSALRE
82 CDK6/CycD1 CDK6, PLSTIRE, MGC59692
83 CDK6/CycD2 CDK6, PLSTIRE
84 CDK6/CycD3 CDK6, PLSTIRE
85 CDK7/CycH/MAT1 CDK7, CAK1, CDKN7, STK1, p39MO15
86 CDK8/CycC CDK8, K35
87 CDK9/CycK CDK9, C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase
88 CDK9/CycT1 CDK9, C-2k, CDC2L4K35, PITALRE, TAK
89 CHK1 CHEK1, n/a
90 CHK2 CHEK2, CDS1, HuCds1, PP1425, RAD53, bA444G7
91 CK1-alpha1 CSNK1A1, CK1, HLCDGP1, PRO2975
92 CK1-delta CSNK1D, HCKID
93 CK1-epsilon CSNK1E, CKIe, HCKIE, MGC10398
94 CK1-gamma1 CSNK1G1
95 CK1-gamma2 CSNK1G2, CK1g2
96 CK1-gamma3 CSNK1G3
97 CK2-alpha1 CSNK2A1, CKII, CK2A1
98 CK2-alpha2 CSNK2A2, n/a
99 CLK1 CLK1, CLK, CLK/STY
100 CLK2 CLK2, MGC61500, clk2, hCLK2
101 CLK3 CLK3, PHCLK3, PHCLK3/152
102 CLK4 CLK4, DKFZp686A20267, CDC-like kinase 4
103 COT MAP3K8, EST, ESTF, TPL2, Tpl-2, c-COT
104 CSF1-R CSF1R, C-FMS, CD115, CSF-1-R, CSFR, FIM2, FMS
105 CSK CSK, n/a
106 DAPK1 DAPK1, n/a
107 DAPK2 DAPK2, DRP-1
108 DAPK3 DAPK3, ZIP, ZIPK
109 DCAMKL2 DCLK2, DCLK, KIAA0369
110 DDR2 N456S DDR2, MIG20a, NTRKR3, TKT, TYRO10
111 DDR2 T654M DDR2, MIG20a, NTRKR3, TKT, TYRO10
112 DDR2 wt DDR2, MIG20a, NTRKR3, TKT, TYRO10
113 DMPK DMPK, DM, DM1, DM1PK, DMK
114 DNA-PK PRKDC, DNAPK, DNPK1, HYRC, HYRC1, XRCC7, p350
115 DYRK1A DYRK1A, DYRK, DYRK1, HP86, MNB, MNBH
116 DYRK1B DYRK1B, MIRK
117 DYRK2 DYRK2
118 DYRK3 DYRK3, DYRK5, RED, REDK
119 DYRK4 DYRK4
120 EEF2K EEF2K, HSU93850, MGC45041, eEF-2K
121 EGF-R d746-750 EGFR, ERBB, mENA, ERBB1
122 EGF-R d747-749/A750P EGFR, ERBB, mENA, ERBB1
123 EGF-R d747-752/P753S EGFR, ERBB, mENA, ERBB1
124 EGF-R d752-759 EGFR, ERBB, mENA, ERBB1
125 EGF-R G719C EGFR, ERBB, mENA, ERBB1
126 EGF-R G719S EGFR, ERBB, mENA, ERBB1
127 EGF-R L858R EGFR, ERBB, ERBB1
128 EGF-R L861Q EGFR, ERBB, mENA, ERBB1
129 EGF-R T790M EGFR, ERBB, ERBB1
130 EGF-R T790M/L858R EGFR, ERBB, ERBB1
131 EGF-R wt EGFR, ERBB, mENA, ERBB1
132 EIF2AK2 EIF2AK2, EIF2AK1, PKR, PRKR
133 EIF2AK3 EIF2AK3, DKFZp781H1925, PEK, PERK, WRS
134 EML4 ALK ALK
135 EML4 ALK F1174L ALK
136 EPHA1 EPHA1, EPH, EPHT, EPHT1
137 EPHA2 EPHA2, ECK
138 EPHA3 EPHA3, ETK, ETK1, EphA3, HEKECK, HEK4, TYRO4
139 EPHA4 EPHA4, HEK8, SEK, TYRO1
140 EPHA5 EPHA5, CEK7, EHK1, EphA5, HEK7, Hek7, TYRO4
141 EPHA6 EPHA6, EHK2, EHK-2, EPA6
142 EPHA7 EPHA7, EHK3, HEK11
143 EPHA8 EPHA8, EEK, EphA8, HEK3, KIAA1459
144 EPHB1 EPHB1, ELK, NET, Hek6, EPHT2
145 EPHB2 EPHB2, DRT, ERK, Hek5, EPHT3, Tyro5
146 EPHB3 EPHB3, ETK2, HEK2, TYRO6
147 EPHB4 EPHB4, HTK, MYK1, TYRO11
148 ERBB2 725YVMA726 ERBB2, CD340, HER2, MLN19, NGL, TKR1
149 ERBB2 wt ERBB2, NEU, NGL, HER2, TKR1, HER-2
150 ERBB4 ERBB4, n/a
151 ERK1 MAPK3, ERT2, HS44KDAP, HUMKER1A, P44ERK1, P44MAPK, PRKM3
152 ERK2 MAPK1, ERK, ERT1, MAPK2, P42MAPK, PRKM1, PRKM2, p38, p40, p41
153 ERK5 MAPK7, BMK1, ERK4, PRKM7
154 ERK7 MAPK15, ERK8, MAPK15
155 FAK aa2-1052 PTK2, FADK, pp125FAK
156 FER FER, TYK3, c-FER, p94-FER
157 FES FES, FPS
158 FGF-R1 V561M FGFR1, FGFR-1, bFGF-R, FLT2, CEK, CD331
159 FGF-R1 wt FGFR1, H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM
160 FGF-R2 FGFR2, FGFR2, BEK, BFR-1, CD332, CEK3, CFD1, ECT1, FGFR-2, JWS, KGFR, KSAM, K-SAM, TK14, TK25
161 FGF-R3 G697C FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
162 FGF-R3 K650E FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
163 FGF-R3 K650M FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
164 FGF-R3 wt FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
165 FGF-R4 FGFR4, TKF, JTK2, MGC20292
166 FGR FGR, SRC2, c-fgr, p55c-fgr
167 FLT3 D835Y FLT3, CD135, FLK2, STK-1, STK1
168 FLT3 ITD FLT3, CD135, FLK2, STK-1, STK1
169 FLT3 wt FLT3, CD135, FLK2, STK-1, STK1
170 FRK FRK, GTK, PTK5, RAK
171 FYN wt FYN, SLK, SYN, p59-Fyn
172 FYN Y531F FYN, SLK, SYN, p59-FYN, cFYN
173 GRK2 ADRBK1
174 GRK3 ADRBK2
175 GRK4 GRK4, GPRK2L, GPRK4, GRK4a, IT11
176 GRK5 GRK5
177 GRK6 GRK6
178 GRK7 GRK7
179 GSG2 GSG2, Haspin
180 GSK3-alpha GSK3A
181 GSK3-beta GSK3B
182 HCK HCK, JTK9
183 HIPK1 HIPK1, KIAA0630, MGC26642, MGC33446, MGC33548, Myak, Nbak2
184 HIPK2 HIPK2, PRO0593
185 HIPK3 HIPK3, ANPK, DYRK6, FIST, FIST3, PKY, YAK1
186 HIPK4 HIPK4, FLJ32818
187 HRI EIF2AK1, HCR
188 IGF1-R IGF1R, JTK13
189 IKK-alpha CHUK, IKBKA, IKK1, IKKA, NFKBIKA, TCF16
190 IKK-beta IKBKB, IKK2, IKKB, NFKBIKB
191 IKK-epsilon IKBKE, IKKE, IKKI, IKK-i, KIAA0151
192 INS-R INSR, n/a
193 INSR-R INSRR, IRR
194 IRAK1 IRAK1, IRAK, Pelle
195 IRAK4 (untagged) IRAK4, REN64, NY-REN-64
196 ITK ITK, EMT 2, LYK 2, PSCTK2 2, IL2-inducible T-cell kinase
197 JAK1 aa583-1154 S729C JAK1, JAK1A, JAK1B, JTK3
198 JAK1 aa583-1154 wt JAK1, JAK1A, JAK1B, JTK3
199 JAK2 JAK2, n/a
200 JAK3 JAK3, JAKL, L-JAK, LJAK
201 JNK1 MAPK8, PRKM8, SAPK1, JNK1-alpha1
202 JNK2 MAPK9, PRKM9, p54aSAPK, JNK2-alpha2
203 JNK3 MAPK10, JNK3A, p54bSAPK
204 KIT A829P KIT, C-Kit, PBT, CD117, SCFR, c-kit
205 KIT D816H KIT, C-Kit, PBT, CD117, SCFR, c-kit
206 KIT D816V KIT, C-Kit, PBT, CD117, SCFR, c-kit
207 KIT T670I KIT, CD117, SCFR, PBT, C-Kit
208 KIT V559D KIT, C-Kit, PBT, CD117, SCFR, c-kit
209 KIT V559D/T670I KIT, C-Kit, PBT, CD117, SCFR, c-kit
210 KIT V559D/V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
211 KIT V560G KIT, C-Kit, PBT, CD117, SCFR, c-kit
212 KIT V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
213 KIT wt KIT, C-Kit, PBT, CD117, SCFR, c-kit
214 LCK LCK, n/a
215 LIMK1 LIMK1, LIMK
216 LIMK2 LIMK2
217 LRRK2 G2019S LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
218 LRRK2 I2020T LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
219 LRRK2 R1441C LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
220 LRRK2 wt LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
221 LTK LTK, TYK1
222 LYN LYN, JTK8
223 MAP3K1 MAP3K1, MAPKKK1, MEKK, MEKK1
224 MAP3K10 MAP3K10, MLK2, MST, MEKK10
225 MAP3K11 MAP3K11, MGC17114, MLK-3, PTK1, SPRK
226 MAP3K7/MAP3K7IP1 MAP3K7, TAK1, TGF1a, MEKK7
227 MAP3K9 MAP3K9, MLK1, PRKE1, MEKK9
228 MAP4K2 MAP4K2, BL44, GCK, RAB8IP
229 MAP4K4 MAP4K4, HGK, MEKKK4, NIK
230 MAP4K5 MAP4K5, KHS1, GCKR, KHS, MAPKKKK5
231 MAPKAPK2 MAPKAPK2, n/a
232 MAPKAPK3 MAPKAPK3, 3PK, MAPKAP, MAPKAP3
233 MAPKAPK5 MAPKAPK5, PRAK
234 MARK1 MARK1, KIAA1477
235 MARK2 MARK2, EMK1, MGC99619, PAR-1, ELKL motif kinase 1
236 MARK3 MARK3, CTAK1, KP78, PAR1A
237 MARK4 MARK4, KIAA1860, MARKL1
238 MASTL MASTL, GLW, GREATWALL, GWL, hGWL, MAST-L, THC2
239 MATK MATK, CHK, CTK, DKFZp434N1212, HHYLTK, HYL, Lsk, MGC1708, MGC2101
240 MEK1 F53L MAP2K1, MAP2K1, MAPKK1, MAPKK 1, MKK1, PRKMK1
241 MEK1 wt MAP2K1, MAPKK1, MKK1, PRKMK1
242 MEK2 MAP2K2, MAPKK2, MKK2, PRKMK2
243 MEK5 MAP2K5, MAP2K5, MAPKK5, MKK5, PRKMK5
244 MEKK2 MAP3K2, MAPKKK2, MEKK2B
245 MEKK3 MAP3K3, MAPKKK3, MEK kinase3
246 MELK MELK, PK38
247 MERTK MERTK, MER, MER-PEN, RP38
248 MET D1228H MET, HGFR, RCCP2
249 MET D1228N MET, HGFR, RCCP2
250 MET F1200I MET, HGFR, RCCP2
251 MET L1195V MET, HGFR, RCCP2
252 MET M1250T MET, HGFR, RCCP2
253 MET wt MET, HGFR, RCCP2
254 MET Y1230A MET, HGFR, RCCP2
255 MET Y1230C MET, HGFR, RCCP2
256 MET Y1230D MET, HGFR, RCCP2
257 MET Y1230H MET, HGFR, RCCP2
258 MET Y1235D MET, HGFR, RCCP2
259 MINK1 MINK1, B55, YSK2, MAP4K6, ZC3
260 MKK4 MAP2K4, JNKK, JNKK1, MAPKK4, MEK4, PRKMK4, SEK, SERK1
261 MKK6 S207D/T211D MAP2K6, MAPKK6, MEK6, MKK6, PRKMK6, SAPKK3
262 MKK7 MAP2K7, MAPKK7, MEK7, PRKMK7
263 MKNK1 MKNK1, MNK1
264 MKNK2 MKNK2, MNK2, GPRK7
265 MLK4 n/a, KIAA1804
266 MST1 STK4, KRS2, YSK3
267 MST2 STK3, MST-2, KRS1
268 MST3 STK24, MST-3, MST3B, STK3
269 MST4 MST4, MASK
270 mTOR FRAP1, FRAP, FRAP2, RAFT1, RAPT1, rapamycin target protein
271 MUSK MUSK, n/a
272 MYLK MYLK, smMLCK, FLJ12216, KRP, MLCK, MLCK108, MLCK210
273 MYLK2 MYLK2, KMLC, MLCK, skMLCK
274 MYLK3 MYLK3, caMLCK, MLCK2, MYLK2
275 NEK1 NEK1, NY-REN-55
276 NEK11 NEK11, FLJ23495
277 NEK2 NEK2, NLK1, HsPK21, HsPK 21
278 NEK3 NEK3, HSPK36, MGC29949
279 NEK4 NEK4, NRK2, STK2
280 NEK6 NEK6, SID6-1512
281 NEK7 NEK7, n/a
282 NEK9 NEK9, DKFZp434D0935, MGC16714, NERCC, NERCC1, Nek8
283 NIK MAP3K14, FTDCR1B, HS, HSNIK
284 NLK NLK, n/a
285 NPM1 ALK n/a, n/a
286 NPM1 ALK F1174L n/a, n/a
287 p38-alpha MAPK14, p38-alpha
288 p38-beta MAPK11, p38-beta
289 p38-delta MAPK13, n/a
290 p38-gamma MAPK12, ERK-6, ERK3, ERK5, ERK6, PRKM12, SAPK-3, SAPK3
291 PAK1 PAK1, PAKalpha
292 PAK2 PAK2, PAK65, PAKgamma
293 PAK3 PAK3, CDKN1A, MRX30, OPHN3, PAK3beta, bPAK, hPAK3
294 PAK4 PAK4, n/a
295 PAK6 PAK6, PAK5
296 PAK7 PAK7, KIAA1264, MGC26232
297 PASK PASK, DKFZP434O051, DKFZp686P2031, KIAA0135, PASKIN, STK3
298 PBK PBK, TOPK, SPK, Nori-3, FLJ14385
299 PDGFR-alpha D842V PDGFRA, PDGFR2, CD140a
300 PDGFR-alpha T674I PDGFRA, PDGFR2, CD140a
301 PDGFR-alpha V561D PDGFRA, PDGFR2, CD140a
302 PDGFR-alpha wt PDGFRA, PDGFR2, CD140a
303 PDGFR-beta PDGFRB, JTK12, PDGFR, CD140B, PDGFR1, PDGF-R-beta
304 PDK1 PDPK1, PKB-like
305 PHKG1 PHKG1, PHKg1
306 PHKG2 PHKG2, PHKg2
307 PI4K2A PI4K2A, PI4KII, PIK42A, RP11-548K23.6
308 PI4K2B PI4K2B, PI4KIIB, PI4KII-BETA, PIK42B
309 PI4KB PI4KB, NPIK, pi4K92, PI4K92, PI4Kbeta, PI4KBETA, PI4K-beta, PI4K-BETA, PI4KIIIBETA, PIK4CB
310 PIK3C2A PIK3C2A, CPK, MGC142218, PI3-K-C2A
311 PIK3C2B PIK3C2B, C2-PI3K, PI3K-C2beta
312 PIK3C2G PIK3C2G, PI3K-C2GAMMA, PI3K-C2-gamma
313 PIK3C3 PIK3C3, hVps34, MGC61518, PI3-kinase type 3, PI3K type 3, Vps34, VPS34
314 PIK3CA/PIK3R1 PIK3CA, MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha
315 PIK3CB D1067A/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
316 PIK3CB D1067V/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
317 PIK3CB D1067Y/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
318 PIK3CB E1051K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
319 PIK3CB E633K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
320 PIK3CB L1049R/PIK3R1 PIK3CB
321 PIK3CB wt/PIK3R1 PIK3CB, PI3K, PI3KBETA, PI3K-beta, PIK3C1, p110-beta
322 PIK3CD/PIK3R1 PIK3CD, p110D, P110DELTA, PI3K, PI3K-delta, p110-delta
323 PIK3CG PIK3CG, p120-PI3K, PI3CG, PI3K, PI3Kgamma, PI3K-gamma, p110-gamma
324 PIM1 PIM1, PIM
325 PIM2 PIM2, n/a
326 PIM3 PIM3, n/a
327 PIP5K1A PIP5K1A, PIP5K1-alpha, PIP5KIalpha, PtdIns(4)P-5-kinase 1 alpha
328 PIP5K1B PIP5K1B, MSS4, PIP5K1-beta, STM7
329 PIP5K1C PIP5K1C, PIP5K1-gamma, PIP5Kgamma, PIP5K-GAMMA, PIPKIg_v4
330 PKA PRKACA, MGC48865, PKA
331 PKC-alpha PRKCA, PKCA, PRKACA, PKC-alpha
332 PKC-beta1 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
333 PKC-beta2 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
334 PKC-delta PRKCD, MAY1, MGC49908, nPKC-delta
335 PKC-epsilon PRKCE, PKCE, nPKC-epsilon
336 PKC-eta PRKCH, PKC-L, PKCL, PRKCL, nPKC-eta
337 PKC-gamma PRKCG, PKCC, PKCG, SCA14, MGC57564
338 PKC-iota PRKCI, PKCI, DXS1179E, MGC26534, nPKC-iota
339 PKC-mu PRKD1, PKD, PKCM, PKC-MU
340 PKC-nu PRKD3, EPK2
341 PKC-theta PRKCQ, PRKCT, nPKC-theta
342 PKC-zeta PRKCZ, PKC2
343 PKC-zeta wt aa184-592 (PKM-zeta) PRKCZ, PKM-zeta, nPKC-zeta, PKC2
344 PKMYT1 PKMYT1, MYT1
345 PKN3 PKN3, PKNbeta, RP11-545E17.1
346 PLK1 PLK1, PLK, STPK13
347 PLK3 PLK3, CNK, FNK, PRK
348 PRK1 PKN1, DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204
349 PRK2 PKN2, PRKCL2, PAK-2
350 PRKD2 PRKD2, PKD2, HSPC187
351 PRKG1 PRKG1, PKG1, CGKI, MGC71944, PGK, PRKG1B, PRKGR1B, cGKIBETA, cGKI-alph
352 PRKG2 PRKG2, PKG2, PRKGR2, cGKII
353 PRKX PRKX, PKX1
354 PYK2 PTK2B, CADTK, CAKB, FADK2, FAK2, PKB, PTK, PYK2, RAFTK, CAK beta
355 RAF1 Y340D/Y341D (untagged) RAF1, c-RAF
356 RET E762Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
357 RET G691S RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
358 RET M918T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
359 RET R749T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
360 RET R813Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
361 RET S891A RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
362 RET V804E RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
363 RET V804L RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
364 RET V804M RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
365 RET wt RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
366 RET Y791F RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
367 RET Y806H RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
368 RIPK2 RIPK2, CARD3, CARDIAK, CCK, GIG30, RICK, RIP-2, RIP2
369 RIPK4 RIPK4, ANKK2, ANKRD3, DIK, MGC129992, MGC129993, PKK, RIP4
370 RIPK5 DSTYK, SgK496, SHIK
371 ROCK1 ROCK1, P160ROCK
372 ROCK2 ROCK2, KIAA0619, ROC2
373 RON MST1R, CD136, CDw136, PTK8
374 ROS ROS1, MCF3
375 RPS6KA1 RPS6KA1, RSK3, HU-1, MAPKAPK1A, RSK, RSK1
376 RPS6KA2 RPS6KA2, RSK1, HU-2, MAPKAPK1C, RSK, RSK3
377 RPS6KA3 RPS6KA3, HU-2, HU-3, ISPK-1, MAPKAPK1B, MRX19, RSK, RSK2
378 RPS6KA4 RPS6KA4, MSK2, RSK-B
379 RPS6KA5 RPS6KA5, MSK1, EC 2.7.11, MGC1911, MSPK1, RLPK, RSKL
380 RPS6KA6 RPS6KA6, RSK4
381 S6K RPS6KB1, S6K1, STK14A
382 S6K-beta RPS6KB2, KLS, P70-beta-1, P70-beta-2, S6K-beta2, S6K2, SRK, p70S6Kb
383 SAK PLK4, SAK, STK18
384 SGK1 SGK, n/a
385 SGK2 SGK2, H-SGK2, dJ138B7.2
386 SGK3 SGKL, CISK, SGK2, SGK3
387 SIK1 SIK1, MSK, SNF1LK, SIK, SIK-1, SNF1LK
388 SIK2 SIK2, QIK, SNF1LK2
389 SIK3 SIK3, L19, QSK, SIK-3
390 SLK SLK, KIAA0204, STK2, bA16H23.1, se20-9
391 SNARK NUAK2, DKFZp434J037
392 SNK PLK2, SNK
393 SRC (GST-HIS-tag) SRC, ASV, SRC1, c-SRC, p60-Src
394 SRMS SRMS, C20orf148, SRM, dJ697K14.1
395 SRPK1 SRPK1, SFRSK1
396 SRPK2 SRPK2, SFRSK2
397 STK17A STK17A, DRAK1
398 STK23 SRPK3, MSSK1, MGC102944
399 STK25 STK25, DKFZp686J1430, SOK1, YSK1
400 STK33 STK33
401 STK39 STK39, STLK3, DCHT, SPAK
402 SYK aa1-635 SYK, n/a
403 TAOK2 TAOK2, KIAA0881, MAP3K17, PSK, PSK1, TAO1, TAO2
404 TAOK3 TAOK3, DPK, JIK, MAP3K18, TAO kinase 3
405 TBK1 TBK1, CDC37, HSPCA, HSPCB, IKBKG, NAK, T2K, TANK, TRAF2
406 TEC TEC, PSCTK4
407 TGFB-R1 TGFBR1, ALK5, ACVRLK4
408 TGFB-R2 TGFBR2, HNPCC6, MFS2, RIIC, TGFR-2, TGFbeta-RII
409 TIE2 R849W TEK, VMCM, TIE-2, VMCM1, CD202B
410 TIE2 wt TEK, VMCM, TIE-2, VMCM1, CD202B
411 TIE2 Y1108F TEK, VMCM, TIE-2, VMCM1, CD202B
412 TIE2 Y897S TEK, VMCM, TIE-2, VMCM1, CD202B
413 TLK1 TLK1, PKU-beta, KIAA0137
414 TLK2 TLK2, MGC44450, PKU-ALPHA
415 TNK1 TNK1, n/a
416 TRK-A G667C MTC, TRK1, TRKA
417 TRK-A wt NTRK1, MTC, TRK, TRK1, TRKA
418 TRK-B NTRK2, GP145-TrkB, TRKB, Trk-B
419 TRK-C NTRK3, GP145-TrkC, TRKC, Trk-C
420 TSF1 STK16, KRCT, MPSK, PKL12
421 TSK2 TSSK2, DGS-G, SPOGA2, FLJ38613
422 TSSK1 TSSK1, FKSG81, SPOGA4, STK22D
423 TTBK1 TTBK1, BDTK
424 TTBK2 TTBK2, BDTK, KIAA1855, RP3-330M21.4
425 TTK TTK, ESK, MPS1L1, PYT
426 TXK TXK, BTKL, PSCTK5, PTK4, RLK
427 TYK2 TYK2, JTK1
428 TYRO3 TYRO3, BYK, Brt, Dtk, Sky, Tif
429 ULK2 ULK2, ATG1B, KIAA0623, Unc51.2
430 VEGF-R1 FLT1, FLT, VEGFR1
431 VEGF-R2 KDR, FLK1, VEGFR, VEGFR2
432 VEGF-R3 FLT4, PCL, VEGFR3
433 VRK1 VRK1, n/a
434 VRK2 VRK2, n/a
435 WEE1 WEE1, WEE1hu
436 WNK1 WNK1, KDP, KIAA0344, PHA2C, PRKWNK1
437 WNK2 WNK2, KIAA1760, NY-CO-43, P/OKcl.13, PRKWNK2, SDCCAG43
438 WNK3 WNK3, KIAA1566, PRKWNK3
439 YES YES, C-YES, HsT441, P61-YES
440 ZAK MLTK, mlklak, AZK
441 ZAP70 ZAP70, SRK, STD, TZK, ZAP-70

Infos in Brief

Kinase Panel

441 kinases, including 89 disease-relevant kinase
mutants and 20 lipid kinases

Assay Technologies

Protein kinases: FlashPlate™-based radiometric assay;
lipid kinases: ADP-Glo™ assay technology (Promega)

ATP conc

App. ATP-Km for each kinase

Testing Modes

Single concentration measurement or IC50 profiling
(10 conc in semi-log steps)

Cpd Submission

100 x Stock solution in 100% DMSO or
pre-weighed powder (request guidelines)

Report

Detailed report for each project

Turnaround Time

No fixed time slots; first come - first served;
routinely within 10 working days

Info Sheets

Method: Radiometric Assay, Method: ATP-Glo™ Assay

List of Kinases for this Service

PDF

Guidelines for Cpd Submission

Guidelines       SPF       CSF