Biochemical Assay Services

Free Choice Kinase Assay Projects

Field of Application

Free choice kinase assay projects allow characterization of your test com-pounds in a self-selected panel of biochemical kinase activity assays. For each project you can freely define (i) the number of test compounds, (ii) the kinase panel, (iii) and the number of data points for each test compound (i.e. number of concentrations and replicates).

Our Products

Number Kinase Synonyms
1 ABL1 E255K ABL1, c-Abl, JTK7, p150
2 ABL1 F317I ABL1, ABL, JTK7, p150, c-ABL, v-abl
3 ABL1 G250E ABL1, ABL, JTK7, p150, c-ABL, v-abl
4 ABL1 H396P ABL1, ABL, JTK7, p150, c-ABL, v-abl
5 ABL1 M351T ABL1, ABL, JTK7, p150, c-ABL, v-abl
6 ABL1 Q252H ABL1, ABL, JTK7, p150, c-ABL, v-abl
7 ABL1 T315I ABL1, ABL, JTK7, p150, c-ABL, v-abl
8 ABL1 wt ABL1, ABL, JTK7, p150, c-ABL, v-abl
9 ABL1 Y253F ABL1, ABL, JTK7, p150, c-ABL, v-abl
10 ABL2 ABL2, ABLL, ARG
11 ACK1 TNK2, ACK, p21cdc42Hs, Activated CDC42 kinase 1
12 ACV-R1 ACVR1, ACTRI, ACVRLK2, ALK2, SKR1
13 ACV-R1B ACVR1B, ACTRIB, ACVRLK4, ALK4, SKR2
14 ACV-R2A ACVR2, ACTRII
15 ACV-R2B ActR-IIB, ACTRIIB
16 ACV-RL1 ACVRL1, ACVRLK1, ALK-1, ALK1, HHT, HHT2, ORW2, SKR3
17 AKT1 aa1-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
18 AKT1 aa106-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
19 AKT2 aa107-481 AKT2, PRKBB, PKBBETA, RAC-BETA
20 AKT3 aa106-479 AKT3, PKBG, PRKBG, STK-2, RAC-gamma, RAC-PK-gamma
21 ALK C1156Y (GST-HIS-tag) ALK, CD246, NBLST3
22 ALK F1174L (GST-HIS-tag) ALK, CD246, NBLST3
23 ALK F1174S (GST-HIS-tag) ALK, CD246, NBLST3
24 ALK G1202R (GST-HIS-tag) ALK, CD246, NBLST3
25 ALK L1196M (GST-HIS-tag) ALK, CD246, NBLST3
26 ALK R1275Q (GST-HIS-tag) ALK, CD246, NBLST3
27 ALK wt (GST-HIS-tag) ALK, CD246, NBLST3
28 AMPK-alpha1 aa1-550 PRKAA1, MGC33776, MGC57364
29 ARK5 NUAK1, KIAA0537
30 ASK1 MAP3K5, ASK1, MAPKKK5, MEKK5
31 Aurora-A STK6, AIK, ARK1, AURA, BTAK, STK15, MGC34538
32 Aurora-B AURKB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AIM-1, STK12
33 Aurora-C AURKC, AIE2, AIK3, STK13
34 AXL AXL, EC, UFO
35 B-RAF V600E BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
36 B-RAF wt BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
37 BLK BLK, n/a
38 BMPR1A BMPR1A, ACVRLK3, ALK3
39 BMX BMX, ETK, PSCTK2, PSCTK3
40 BRK PTK6, n/a
41 BRSK1 BRSK1, KIAA1811
42 BRSK2 C11orf7, FLJ41362, HUSSY-12, PEN11B, SAD1, STK29
43 BTK BTK, AGMX1, AT, ATK, BPK, PSCTK1
44 BUB1B BUB1B, BUBR1, Bub1A, MAD3L, hBUBR1
45 CAMK1D CAMK1D, CKLiK, CaM-K1, CaMKID
46 CAMK2A CAMK2A, CAMKA, KIAA0968
47 CAMK2B CAMK2B, CAM2, CAMK2, CAMKB, MGC29528
48 CAMK2D CAMK2D, CAMKD, MGC44911, CaMKII delta
49 CAMK2G CAMK2G, CAMK, CAMK-II, CAMKG, MGC26678
50 CAMK4 CAMK4, CaMK-GR, MGC36771
51 CAMKK1 CAMKK1, CAMKKA, DKFZp761M0423, MGC34095
52 CAMKK2 CAMKK2, CAMKK, CAMKKB, KIAA0787, MGC15254
53 CCDC6-RET CCDC6-RET, CCDC6-RETa
54 CDC42BPA CDC42BPA, MRCK-alpha
55 CDC42BPB CDC42BPB, MRCK-beta, MRCKb
56 CDC7/DBF4 CDC7, CDC7L1, HsCdc7, HsCDC7, Hsk1, huCdc7
57 CDK1/CycA2 CDC2, p34
58 CDK1/CycB1 CDC2, p34
59 CDK1/CycE1 CDC2, p34
60 CDK12 R722C/CycK CDK12, CRKRS, CRK7
61 CDK12 wt/CycK CDK12, CRKRS, CRK7
62 CDK13/CycK CDK13, CDC2L, CDC2L5, CHED
63 CDK16/CycY CDK16, PCTAIRE1, PCTAIRE, PCTGAIRE, PCTK1
64 CDK17/p35NCK CDK17, PCTAIRE2, PCTK2
65 CDK18/CycY CDK18, PCTAIRE, PCTAIRE3, PCTK3
66 CDK19/CycC CDK19, CDC2L6, CDK11
67 CDK2/CycA2 CDK2, p33(CDK2)
68 CDK2/CycD1 CDK2, p33
69 CDK2/CycE1 CDK2, p33(CDK2)
70 CDK20/CycH CDK20, CAK-kinase p42
71 CDK20/CycT1 CDK20, CAK-kinase p42, CCRK, CDCH, p42, PNQALRE
72 CDK3/CycC CDK3, CDKN3
73 CDK3/CycE1 CDK3, n/a
74 CDK4/CycD1 CDK4, CMM3, PSK-J3, MGC14458
75 CDK4/CycD2 CDK4, CMM3, PSK-J3
76 CDK4/CycD3 CDK4, CMM3, PSK-J3, MGC14458
77 CDK5/p25NCK CDK5, PSSALRE
78 CDK5/p35NCK CDK5, PSSALRE
79 CDK6/CycD1 CDK6, PLSTIRE, MGC59692
80 CDK6/CycD2 CDK6, PLSTIRE
81 CDK6/CycD3 CDK6, PLSTIRE
82 CDK7/CycH/MAT1 CDK7, CAK1, CDKN7, STK1, p39MO15
83 CDK8/CycC CDK8, K35
84 CDK9/CycK CDK9, C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase
85 CDK9/CycT1 CDK9, C-2k, CDC2L4K35, PITALRE, TAK
86 CHK1 CHEK1, n/a
87 CHK2 CHEK2, CDS1, HuCds1, PP1425, RAD53, bA444G7
88 CK1-alpha1 CSNK1A1, CK1, HLCDGP1, PRO2975
89 CK1-delta CSNK1D, HCKID
90 CK1-epsilon CSNK1E, CKIe, HCKIE, MGC10398
91 CK1-gamma1 CSNK1G1
92 CK1-gamma2 CSNK1G2, CK1g2
93 CK1-gamma3 CSNK1G3
94 CK2-alpha1 CSNK2A1, CKII, CK2A1
95 CK2-alpha2 CSNK2A2, n/a
96 CLK1 CLK1, CLK, CLK/STY
97 CLK2 CLK2, MGC61500, clk2, hCLK2
98 CLK3 CLK3, PHCLK3, PHCLK3/152
99 CLK4 CLK4, DKFZp686A20267, CDC-like kinase 4
100 COT MAP3K8, EST, ESTF, TPL2, Tpl-2, c-COT
101 CSF1-R CSF1R, C-FMS, CD115, CSF-1-R, CSFR, FIM2, FMS
102 CSK CSK, n/a
103 DAPK1 DAPK1, n/a
104 DAPK2 DAPK2, DRP-1
105 DAPK3 DAPK3, ZIP, ZIPK
106 DCAMKL2 DCLK2, DCLK, KIAA0369
107 DDR2 N456S DDR2, MIG20a, NTRKR3, TKT, TYRO10
108 DDR2 T654M DDR2, MIG20a, NTRKR3, TKT, TYRO10
109 DDR2 wt DDR2, MIG20a, NTRKR3, TKT, TYRO10
110 DMPK DMPK, DM, DM1, DM1PK, DMK
111 DNA-PK PRKDC, DNAPK, DNPK1, HYRC, HYRC1, XRCC7, p350
112 DYRK1A DYRK1A, DYRK, DYRK1, HP86, MNB, MNBH
113 DYRK1B DYRK1B, MIRK
114 DYRK2 DYRK2
115 DYRK3 DYRK3, DYRK5, RED, REDK
116 DYRK4 DYRK4
117 EEF2K EEF2K, HSU93850, MGC45041, eEF-2K
118 EGF-R d746-750 EGFR, ERBB, mENA, ERBB1
119 EGF-R d747-749/A750P EGFR, ERBB, mENA, ERBB1
120 EGF-R d747-752/P753S EGFR, ERBB, mENA, ERBB1
121 EGF-R d752-759 EGFR, ERBB, mENA, ERBB1
122 EGF-R G719C EGFR, ERBB, mENA, ERBB1
123 EGF-R G719S EGFR, ERBB, mENA, ERBB1
124 EGF-R L858R EGFR, ERBB, ERBB1
125 EGF-R L861Q EGFR, ERBB, mENA, ERBB1
126 EGF-R T790M EGFR, ERBB, ERBB1
127 EGF-R T790M/L858R EGFR, ERBB, ERBB1
128 EGF-R wt EGFR, ERBB, mENA, ERBB1
129 EIF2AK2 EIF2AK2, EIF2AK1, PKR, PRKR
130 EIF2AK3 EIF2AK3, DKFZp781H1925, PEK, PERK, WRS
131 EML4 ALK ALK
132 EML4 ALK F1174L ALK
133 EPHA1 EPHA1, EPH, EPHT, EPHT1
134 EPHA2 EPHA2, ECK
135 EPHA3 EPHA3, ETK, ETK1, EphA3, HEKECK, HEK4, TYRO4
136 EPHA4 EPHA4, HEK8, SEK, TYRO1
137 EPHA5 EPHA5, CEK7, EHK1, EphA5, HEK7, Hek7, TYRO4
138 EPHA6 EPHA6, EHK2, EHK-2, EPA6
139 EPHA7 EPHA7, EHK3, HEK11
140 EPHA8 EPHA8, EEK, EphA8, HEK3, KIAA1459
141 EPHB1 EPHB1, ELK, NET, Hek6, EPHT2
142 EPHB2 EPHB2, DRT, ERK, Hek5, EPHT3, Tyro5
143 EPHB3 EPHB3, ETK2, HEK2, TYRO6
144 EPHB4 EPHB4, HTK, MYK1, TYRO11
145 ERBB2 725YVMA726 ERBB2, CD340, HER2, MLN19, NGL, TKR1
146 ERBB2 wt ERBB2, NEU, NGL, HER2, TKR1, HER-2
147 ERBB4 ERBB4, n/a
148 ERK1 MAPK3, ERT2, HS44KDAP, HUMKER1A, P44ERK1, P44MAPK, PRKM3
149 ERK2 MAPK1, ERK, ERT1, MAPK2, P42MAPK, PRKM1, PRKM2, p38, p40, p41
150 ERK5 MAPK7, BMK1, ERK4, PRKM7
151 ERK7 MAPK15, ERK8, MAPK15
152 FAK aa2-1052 PTK2, FADK, pp125FAK
153 FER FER, TYK3, c-FER, p94-FER
154 FES FES, FPS
155 FGF-R1 V561M FGFR1, FGFR-1, bFGF-R, FLT2, CEK, CD331
156 FGF-R1 wt FGFR1, H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM
157 FGF-R2 FGFR2, FGFR2, BEK, BFR-1, CD332, CEK3, CFD1, ECT1, FGFR-2, JWS, KGFR, KSAM, K-SAM, TK14, TK25
158 FGF-R3 G697C FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
159 FGF-R3 K650E FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
160 FGF-R3 K650M FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
161 FGF-R3 wt FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
162 FGF-R4 FGFR4, TKF, JTK2, MGC20292
163 FGR FGR, SRC2, c-fgr, p55c-fgr
164 FLT3 D835Y FLT3, CD135, FLK2, STK-1, STK1
165 FLT3 ITD FLT3, CD135, FLK2, STK-1, STK1
166 FLT3 wt FLT3, CD135, FLK2, STK-1, STK1
167 FRK FRK, GTK, PTK5, RAK
168 FYN wt FYN, SLK, SYN, p59-Fyn
169 FYN Y531F FYN, SLK, SYN, p59-FYN, cFYN
170 GRK2 ADRBK1
171 GRK3 ADRBK2
172 GRK4 GRK4, GPRK2L, GPRK4, GRK4a, IT11
173 GRK5 GRK5
174 GRK6 GRK6
175 GRK7 GRK7
176 GSG2 GSG2, Haspin
177 GSK3-alpha GSK3A
178 GSK3-beta GSK3B, n/a
179 HCK HCK, JTK9
180 HIPK1 HIPK1, KIAA0630, MGC26642, MGC33446, MGC33548, Myak, Nbak2
181 HIPK2 HIPK2, PRO0593
182 HIPK3 HIPK3, ANPK, DYRK6, FIST, FIST3, PKY, YAK1
183 HIPK4 HIPK4, FLJ32818
184 HRI EIF2AK1, HCR
185 IGF1-R IGF1R, JTK13
186 IKK-alpha CHUK, IKBKA, IKK1, IKKA, NFKBIKA, TCF16
187 IKK-beta IKBKB, IKK2, IKKB, NFKBIKB
188 IKK-epsilon IKBKE, IKKE, IKKI, IKK-i, KIAA0151
189 INS-R INSR, n/a
190 INSR-R INSRR, IRR
191 IRAK1 IRAK1, IRAK, Pelle
192 IRAK4 (untagged) IRAK4, REN64, NY-REN-64
193 ITK ITK, EMT 2, LYK 2, PSCTK2 2, IL2-inducible T-cell kinase
194 JAK1 aa583-1154 S729C JAK1, JAK1A, JAK1B, JTK3
195 JAK1 aa583-1154 wt JAK1, JAK1A, JAK1B, JTK3
196 JAK2 JAK2, n/a
197 JAK3 JAK3, JAKL, L-JAK, LJAK
198 JNK1 MAPK8, PRKM8, SAPK1, JNK1-alpha1
199 JNK2 MAPK9, PRKM9, p54aSAPK, JNK2-alpha2
200 JNK3 MAPK10, JNK3A, p54bSAPK
201 KIT A829P KIT, C-Kit, PBT, CD117, SCFR, c-kit
202 KIT D816H KIT, C-Kit, PBT, CD117, SCFR, c-kit
203 KIT D816V KIT, C-Kit, PBT, CD117, SCFR, c-kit
204 KIT T670I KIT, CD117, SCFR, PBT, C-Kit
205 KIT V559D KIT, C-Kit, PBT, CD117, SCFR, c-kit
206 KIT V559D/T670I KIT, C-Kit, PBT, CD117, SCFR, c-kit
207 KIT V559D/V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
208 KIT V560G KIT, C-Kit, PBT, CD117, SCFR, c-kit
209 KIT V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
210 KIT wt KIT, C-Kit, PBT, CD117, SCFR, c-kit
211 LCK LCK, n/a
212 LIMK1 LIMK1, LIMK
213 LIMK2 LIMK2
214 LRRK2 G2019S LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
215 LRRK2 I2020T LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
216 LRRK2 R1441C LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
217 LRRK2 wt LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
218 LTK LTK, TYK1
219 LYN LYN, JTK8
220 MAP3K1 MAP3K1, MAPKKK1, MEKK, MEKK1
221 MAP3K10 MAP3K10, MLK2, MST, MEKK10
222 MAP3K11 MAP3K11, MGC17114, MLK-3, PTK1, SPRK
223 MAP3K7/MAP3K7IP1 MAP3K7, TAK1, TGF1a, MEKK7
224 MAP3K9 MAP3K9, MLK1, PRKE1, MEKK9
225 MAP4K2 MAP4K2, BL44, GCK, RAB8IP
226 MAP4K4 MAP4K4, HGK, MEKKK4, NIK
227 MAP4K5 MAP4K5, KHS1, GCKR, KHS, MAPKKKK5
228 MAPKAPK2 MAPKAPK2, n/a
229 MAPKAPK3 MAPKAPK3, 3PK, MAPKAP, MAPKAP3
230 MAPKAPK5 MAPKAPK5, PRAK
231 MARK1 MARK1, KIAA1477
232 MARK2 MARK2, EMK1, MGC99619, PAR-1, ELKL motif kinase 1
233 MARK3 MARK3, CTAK1, KP78, PAR1A
234 MARK4 MARK4, KIAA1860, MARKL1
235 MASTL MASTL, GLW, GREATWALL, GWL, hGWL, MAST-L, THC2
236 MATK MATK, CHK, CTK, DKFZp434N1212, HHYLTK, HYL, Lsk, MGC1708, MGC2101
237 MEK1 F53L MAP2K1, MAP2K1, MAPKK1, MAPKK 1, MKK1, PRKMK1
238 MEK1 wt MAP2K1, MAPKK1, MKK1, PRKMK1
239 MEK2 MAP2K2, MAPKK2, MKK2, PRKMK2
240 MEK5 MAP2K5, MAP2K5, MAPKK5, MKK5, PRKMK5
241 MEKK2 MAP3K2, MAPKKK2, MEKK2B
242 MEKK3 MAP3K3, MAPKKK3, MEK kinase3
243 MELK MELK, PK38
244 MERTK MERTK, MER, MER-PEN, RP38
245 MET D1228H MET, HGFR, RCCP2
246 MET D1228N MET, HGFR, RCCP2
247 MET F1200I MET, HGFR, RCCP2
248 MET M1250T MET, HGFR, RCCP2
249 MET wt MET, HGFR, RCCP2
250 MET Y1230A MET, HGFR, RCCP2
251 MET Y1230C MET, HGFR, RCCP2
252 MET Y1230D MET, HGFR, RCCP2
253 MET Y1230H MET, HGFR, RCCP2
254 MET Y1235D MET, HGFR, RCCP2
255 MINK1 MINK1, B55, YSK2, MAP4K6, ZC3
256 MKK4 MAP2K4, JNKK, JNKK1, MAPKK4, MEK4, PRKMK4, SEK, SERK1
257 MKK6 S207D/T211D MAP2K6, MAPKK6, MEK6, MKK6, PRKMK6, SAPKK3
258 MKK7 MAP2K7, MAPKK7, MEK7, PRKMK7
259 MKNK1 MKNK1, MNK1
260 MKNK2 MKNK2, MNK2, GPRK7
261 MLK4 n/a, KIAA1804
262 MST1 STK4, KRS2, YSK3
263 MST2 STK3, MST-2, KRS1
264 MST3 STK24, MST-3, MST3B, STK3
265 MST4 MST4, MASK
266 mTOR FRAP1, FRAP, FRAP2, RAFT1, RAPT1, rapamycin target protein
267 MUSK MUSK, n/a
268 MYLK MYLK, smMLCK, FLJ12216, KRP, MLCK, MLCK108, MLCK210
269 MYLK2 MYLK2, KMLC, MLCK, skMLCK
270 MYLK3 MYLK3, caMLCK, MLCK2, MYLK2
271 NEK1 NEK1, KIAA1901, NY-REN-55
272 NEK11 NEK11, FLJ23495
273 NEK2 NEK2, NLK1, HsPK21, HsPK 21
274 NEK3 NEK3, HSPK36, MGC29949
275 NEK4 NEK4, NRK2, STK2
276 NEK6 NEK6, SID6-1512
277 NEK7 NEK7, n/a
278 NEK9 NEK9, DKFZp434D0935, MGC16714, NERCC, NERCC1, Nek8
279 NIK MAP3K14, FTDCR1B, HS, HSNIK
280 NLK NLK, n/a
281 NPM1 ALK n/a, n/a
282 NPM1 ALK F1174L n/a, n/a
283 p38-alpha MAPK14, p38-alpha
284 p38-beta MAPK11, p38-beta
285 p38-delta MAPK13, n/a
286 p38-gamma MAPK12, ERK-6, ERK3, ERK5, ERK6, PRKM12, SAPK-3, SAPK3
287 PAK1 PAK1, PAKalpha
288 PAK2 PAK2, PAK65, PAKgamma
289 PAK3 PAK3, CDKN1A, MRX30, OPHN3, PAK3beta, bPAK, hPAK3
290 PAK4 PAK4, n/a
291 PAK6 PAK6, PAK5
292 PAK7 PAK7, KIAA1264, MGC26232
293 PASK PASK, DKFZP434O051, DKFZp686P2031, KIAA0135, PASKIN, STK3
294 PBK PBK, TOPK, SPK, Nori-3, FLJ14385
295 PDGFR-alpha D842V PDGFRA, PDGFR2, CD140a
296 PDGFR-alpha T674I PDGFRA, PDGFR2, CD140a
297 PDGFR-alpha V561D PDGFRA, PDGFR2, CD140a
298 PDGFR-alpha wt PDGFRA, PDGFR2, CD140a
299 PDGFR-beta PDGFRB, JTK12, PDGFR, CD140B, PDGFR1, PDGF-R-beta
300 PDK1 PDPK1, PKB-like
301 PHKG1 PHKG1, PHKg1
302 PHKG2 PHKG2, PHKg2
303 PI4K2A PI4K2A, PI4KII, PIK42A, RP11-548K23.6
304 PI4K2B PI4K2B, PI4KIIB, PI4KII-BETA, PIK42B
305 PI4KB PI4KB, NPIK, pi4K92, PI4K92, PI4Kbeta, PI4KBETA, PI4K-beta, PI4K-BETA, PI4KIIIBETA, PIK4CB
306 PIK3C2A PIK3C2A, CPK, MGC142218, PI3-K-C2A
307 PIK3C2B PIK3C2B, C2-PI3K, PI3K-C2beta
308 PIK3C2G PIK3C2G, PI3K-C2GAMMA, PI3K-C2-gamma
309 PIK3C3 PIK3C3, hVps34, MGC61518, PI3-kinase type 3, PI3K type 3, Vps34, VPS34
310 PIK3CA/PIK3R1 PIK3CA, MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha
311 PIK3CB D1067A/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
312 PIK3CB D1067V/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
313 PIK3CB D1067Y/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
314 PIK3CB E1051K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
315 PIK3CB E633K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
316 PIK3CB wt/PIK3R1 PIK3CB, PI3K, PI3KBETA, PI3K-beta, PIK3C1, p110-beta
317 PIK3CD/PIK3R1 PIK3CD, p110D, P110DELTA, PI3K, PI3K-delta, p110-delta
318 PIK3CG PIK3CG, p120-PI3K, PI3CG, PI3K, PI3Kgamma, PI3K-gamma, p110-gamma
319 PIM1 PIM1, PIM
320 PIM2 PIM2, n/a
321 PIM3 PIM3, n/a
322 PIP5K1A PIP5K1A, PIP5K1-alpha, PIP5KIalpha, PtdIns(4)P-5-kinase 1 alpha
323 PIP5K1B PIP5K1B, MSS4, PIP5K1-beta, STM7
324 PIP5K1C PIP5K1C, PIP5K1-gamma, PIP5Kgamma, PIP5K-GAMMA, PIPKIg_v4
325 PKA PRKACA, MGC48865, PKA
326 PKC-alpha PRKCA, PKCA, PRKACA, PKC-alpha
327 PKC-beta1 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
328 PKC-beta2 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
329 PKC-delta PRKCD, MAY1, MGC49908, nPKC-delta
330 PKC-epsilon PRKCE, PKCE, nPKC-epsilon
331 PKC-eta PRKCH, PKC-L, PKCL, PRKCL, nPKC-eta
332 PKC-gamma PRKCG, PKCC, PKCG, SCA14, MGC57564
333 PKC-iota PRKCI, PKCI, DXS1179E, MGC26534, nPKC-iota
334 PKC-mu PRKD1, PKD, PKCM, PKC-MU
335 PKC-nu PRKD3, EPK2
336 PKC-theta PRKCQ, PRKCT, nPKC-theta
337 PKC-zeta PRKCZ, PKC2
338 PKC-zeta wt aa184-592 (PKM-zeta) PRKCZ, PKM-zeta, nPKC-zeta, PKC2
339 PKMYT1 PKMYT1, MYT1
340 PKN3 PKN3, PKNbeta, RP11-545E17.1
341 PLK1 PLK1, PLK, STPK13
342 PLK3 PLK3, CNK, FNK, PRK
343 PRK1 PKN1, DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204
344 PRK2 PKN2, PRKCL2, PAK-2
345 PRKD2 PRKD2, PKD2, HSPC187
346 PRKG1 PRKG1, PKG1, CGKI, MGC71944, PGK, PRKG1B, PRKGR1B, cGKIBETA, cGKI-alph
347 PRKG2 PRKG2, PKG2, PRKGR2, cGKII
348 PRKX PRKX, PKX1
349 PYK2 PTK2B, CADTK, CAKB, FADK2, FAK2, PKB, PTK, PYK2, RAFTK, CAK beta
350 RAF1 Y340D/Y341D (untagged) RAF1, c-RAF
351 RET E762Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
352 RET G691S RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
353 RET M918T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
354 RET R749T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
355 RET R813Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
356 RET S891A RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
357 RET V804E RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
358 RET V804L RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
359 RET V804M RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
360 RET wt RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
361 RET Y791F RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
362 RET Y806H RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
363 RIPK2 RIPK2, CARD3, CARDIAK, CCK, GIG30, RICK, RIP-2, RIP2
364 RIPK4 RIPK4, ANKK2, ANKRD3, DIK, MGC129992, MGC129993, PKK, RIP4
365 RIPK5 DSTYK, SgK496, SHIK
366 ROCK1 ROCK1, P160ROCK
367 ROCK2 ROCK2, KIAA0619, ROC2
368 RON MST1R, CD136, CDw136, PTK8
369 ROS ROS1, MCF3
370 RPS6KA1 RPS6KA1, RSK3, HU-1, MAPKAPK1A, RSK, RSK1
371 RPS6KA2 RPS6KA2, RSK1, HU-2, MAPKAPK1C, RSK, RSK3
372 RPS6KA3 RPS6KA3, HU-2, HU-3, ISPK-1, MAPKAPK1B, MRX19, RSK, RSK2
373 RPS6KA4 RPS6KA4, MSK2, RSK-B
374 RPS6KA5 RPS6KA5, MSK1, EC 2.7.11, MGC1911, MSPK1, RLPK, RSKL
375 RPS6KA6 RPS6KA6, RSK4
376 S6K RPS6KB1, S6K1, STK14A
377 S6K-beta RPS6KB2, KLS, P70-beta-1, P70-beta-2, S6K-beta2, S6K2, SRK, p70S6Kb
378 SAK PLK4, SAK, STK18
379 SGK1 SGK, n/a
380 SGK2 SGK2, H-SGK2, dJ138B7.2
381 SGK3 SGKL, CISK, SGK2, SGK3
382 SIK1 SIK1, MSK, SNF1LK, SIK, SIK-1, SNF1LK
383 SIK2 SIK2, QIK, SNF1LK2
384 SIK3 SIK3, L19, QSK, SIK-3
385 SLK SLK, KIAA0204, STK2, bA16H23.1, se20-9
386 SNARK NUAK2, DKFZp434J037
387 SNK PLK2, SNK
388 SRC (GST-HIS-tag) SRC, ASV, SRC1, c-SRC, p60-Src
389 SRMS SRMS, C20orf148, SRM, dJ697K14.1
390 SRPK1 SRPK1, SFRSK1
391 SRPK2 SRPK2, SFRSK2
392 STK17A STK17A, DRAK1
393 STK23 SRPK3, MSSK1, MGC102944
394 STK25 STK25, DKFZp686J1430, SOK1, YSK1
395 STK33 STK33
396 STK39 STK39, STLK3, DCHT, SPAK
397 SYK aa1-635 SYK, n/a
398 TAOK2 TAOK2, KIAA0881, MAP3K17, PSK, PSK1, TAO1, TAO2
399 TAOK3 TAOK3, DPK, JIK, MAP3K18, TAO kinase 3
400 TBK1 TBK1, CDC37, HSPCA, HSPCB, IKBKG, NAK, T2K, TANK, TRAF2
401 TEC TEC, PSCTK4
402 TGFB-R1 TGFBR1, ALK5, ACVRLK4
403 TGFB-R2 TGFBR2, HNPCC6, MFS2, RIIC, TGFR-2, TGFbeta-RII
404 TIE2 R849W TEK, VMCM, TIE-2, VMCM1, CD202B
405 TIE2 wt TEK, VMCM, TIE-2, VMCM1, CD202B
406 TIE2 Y1108F TEK, VMCM, TIE-2, VMCM1, CD202B
407 TIE2 Y897S TEK, VMCM, TIE-2, VMCM1, CD202B
408 TLK1 TLK1, PKU-beta, KIAA0137
409 TLK2 TLK2, MGC44450, PKU-ALPHA
410 TNK1 TNK1, n/a
411 TRK-A G667C MTC, TRK1, TRKA
412 TRK-A wt NTRK1, MTC, TRK, TRK1, TRKA
413 TRK-B NTRK2, GP145-TrkB, TRKB, Trk-B
414 TRK-C NTRK3, GP145-TrkC, TRKC, Trk-C
415 TSF1 STK16, KRCT, MPSK, PKL12
416 TSK2 TSSK2, DGS-G, SPOGA2, FLJ38613
417 TSSK1 TSSK1, FKSG81, SPOGA4, STK22D
418 TTBK1 TTBK1, BDTK
419 TTBK2 TTBK2, BDTK, KIAA1855, RP3-330M21.4
420 TTK TTK, ESK, MPS1L1, PYT
421 TXK TXK, BTKL, PSCTK5, PTK4, RLK
422 TYK2 TYK2, JTK1
423 TYRO3 TYRO3, BYK, Brt, Dtk, Sky, Tif
424 VEGF-R1 FLT1, FLT, VEGFR1
425 VEGF-R2 KDR, FLK1, VEGFR, VEGFR2
426 VEGF-R3 FLT4, PCL, VEGFR3
427 VRK1 VRK1, n/a
428 VRK2 VRK2, n/a
429 WEE1 WEE1, WEE1hu
430 WNK1 WNK1, KDP, KIAA0344, PHA2C, PRKWNK1
431 WNK2 WNK2, KIAA1760, NY-CO-43, P/OKcl.13, PRKWNK2, SDCCAG43
432 WNK3 WNK3, KIAA1566, PRKWNK3
433 YES YES, C-YES, HsT441, P61-YES
434 ZAK MLTK, mlklak, AZK
435 ZAP70 ZAP70, SRK, STD, TZK, ZAP-70

Infos in Brief

Kinase Panel

435 kinases, including 87 disease-relevant kinase
mutants and 19 lipid kinases

Assay Technologies

Protein kinases: FlashPlate™-based radiometric assay;
lipid kinases: ADP-Glo™ assay technology (Promega)

ATP Conc

App. ATP-Km for each kinase

Testing Modes

Single concentration measurement or IC50 profiling
(10 conc in semi-log steps)

Cpd Submission

100 x Stock solution in 100% DMSO or
pre-weighed powder (request guidelines)

Report

Detailed report for each project

Turnaround Time

No fixed time slots; first come - first served;
routinely within 10 working days

Info Sheets

Method: Radiometric Assay, Method: ATP-Glo™ Assay

List of Kinases for this Service

PDF