Biochemical Assay Services

Free Choice Kinase Assay Projects

Field of Application

Free choice kinase assay projects allow characterization of your test com-pounds in a self-selected panel of biochemical kinase activity assays. For each project you can freely define (i) the number of test compounds, (ii) the kinase panel, (iii) and the number of data points for each test compound (i.e. number of concentrations and replicates).

Our Products

Number Kinase Synonyms
1 ABL1 E255K ABL1, ABL, JTK7, p150, c-ABL, v-abl
2 ABL1 F317I ABL1, ABL, JTK7, p150, c-ABL, v-abl
3 ABL1 G250E ABL1, ABL, JTK7, p150, c-ABL, v-abl
4 ABL1 H396P ABL1, ABL, JTK7, p150, c-ABL, v-abl
5 ABL1 M351T ABL1, ABL, JTK7, p150, c-ABL, v-abl
6 ABL1 Q252H ABL1, ABL, JTK7, p150, c-ABL, v-abl
7 ABL1 T315I ABL1, ABL, JTK7, p150, c-ABL, v-abl
8 ABL1 wt ABL1, ABL, JTK7, p150, c-ABL, v-abl
9 ABL1 Y253F ABL1, ABL, JTK7, p150, c-ABL, v-abl
10 ABL2 ABL2, ARG, ABLL
11 ABL2 ABLL, ARG
12 ACK1 TNK2, ACK, p21cdc42Hs, Activated CDC42 kinase 1
13 ACV-R1 ACVR1, ACTRI, ACVRLK2, ALK2, SKR1
14 ACV-R1B ACVR1B, ACTRIB, ACVRLK4, ALK4, SKR2
15 ACV-R2A ACVR2, ACTRII
16 ACV-R2B ActR-IIB, ACTRIIB
17 ACV-RL1 ACVRL1, ACVRLK1, ALK-1, ALK1, HHT, HHT2, ORW2, SKR3
18 AKT1 aa1-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
19 AKT1 aa106-480 AKT1, PKB, RAC, PRKBA, RAC-ALPHA
20 AKT2 aa107-481 AKT2, PRKBB, PKBBETA, RAC-BETA
21 AKT3 aa106-479 AKT3, PKBG, PRKBG, STK-2, RAC-gamma, RAC-PK-gamma
22 ALK C1156Y (GST-HIS-tag) ALK, CD246, NBLST3
23 ALK F1174L (GST-HIS-tag) ALK, CD246, NBLST3
24 ALK F1174S (GST-HIS-tag) ALK, CD246, NBLST3
25 ALK G1202R (GST-HIS-tag) ALK, CD246, NBLST3
26 ALK L1196M (GST-HIS-tag) ALK, CD246, NBLST3
27 ALK R1275Q (GST-HIS-tag) ALK, CD246, NBLST3
28 ALK wt (GST-HIS-tag) ALK, CD246, NBLST3
29 AMPK-alpha1 aa1-550 PRKAA1, MGC33776, MGC57364
30 ARK5 NUAK1, KIAA0537
31 ASK1 MAP3K5, ASK1, MAPKKK5, MEKK5
32 Aurora-A STK6, AIK, ARK1, AURA, BTAK, STK15, MGC34538
33 Aurora-B AURKB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AIM-1, STK12
34 Aurora-C AURKC, AIE2, AIK3, STK13
35 AXL AXL, EC, UFO
36 B-RAF V600E BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
37 B-RAF wt BRAF, B-Raf, B-raf-1, BRAF1, RAFB1
38 BLK BLK, n/a
39 BMPR1A BMPR1A, ACVRLK3, ALK3
40 BMX BMX, ETK, PSCTK2, PSCTK3
41 BRK PTK6, n/a
42 BRSK1 BRSK1, KIAA1811
43 BRSK2 C11orf7, FLJ41362, HUSSY-12, PEN11B, SAD1, STK29
44 BTK BTK, AGMX1, AT, ATK, BPK, PSCTK1
45 BUB1B BUB1B, BUBR1, Bub1A, MAD3L, hBUBR1
46 CAMK1D CAMK1D, CKLiK, CaM-K1, CaMKID
47 CAMK2A CAMK2A, CAMKA, KIAA0968
48 CAMK2B CAMK2B, CAM2, CAMK2, CAMKB, MGC29528
49 CAMK2D CAMK2D, CAMKD, MGC44911, CaMKII delta
50 CAMK2G CAMK2G, CAMK, CAMK-II, CAMKG, MGC26678
51 CAMK4 CAMK4, CaMK-GR, MGC36771
52 CAMKK1 CAMKK1, CAMKKA, DKFZp761M0423, MGC34095
53 CAMKK2 CAMKK2, CAMKK, CAMKKB, KIAA0787, MGC15254
54 CCDC6-RET CCDC6-RET, CCDC6-RETa
55 CDC42BPA CDC42BPA, MRCK-alpha
56 CDC42BPB CDC42BPB, MRCK-beta, MRCKb
57 CDC7/DBF4 CDC7, CDC7L1, HsCdc7, HsCDC7, Hsk1, huCdc7
58 CDK1/CycA2 CDC2, p34
59 CDK1/CycB1 CDC2, p34
60 CDK1/CycE1 CDC2, p34
61 CDK12 R722C/CycK CDK12, CRKRS, CRK7
62 CDK12 wt/CycK CDK12, CRKRS, CRK7
63 CDK13/CycK CDK13, CDC2L, CDC2L5, CHED
64 CDK16/CycY CDK16, PCTAIRE1, PCTAIRE, PCTGAIRE, PCTK1
65 CDK17/p35NCK CDK17, PCTAIRE2, PCTK2
66 CDK18/CycY CDK18, PCTAIRE, PCTAIRE3, PCTK3
67 CDK19/CycC CDK19, CDC2L6, CDK11
68 CDK2/CycA2 CDK2, p33(CDK2)
69 CDK2/CycD1 CDK2, p33
70 CDK2/CycE1 CDK2, p33(CDK2)
71 CDK20/CycH CDK20, CAK-kinase p42
72 CDK20/CycT1 CDK20, CAK-kinase p42, CCRK, CDCH, p42, PNQALRE
73 CDK3/CycC CDK3, CDKN3
74 CDK3/CycE1 CDK3, n/a
75 CDK4/CycD1 CDK4, CMM3, PSK-J3, MGC14458
76 CDK4/CycD2 CDK4, CMM3, PSK-J3
77 CDK4/CycD3 CDK4, CMM3, PSK-J3, MGC14458
78 CDK5/p25NCK CDK5, PSSALRE
79 CDK5/p35NCK CDK5, PSSALRE
80 CDK6/CycD1 CDK6, PLSTIRE, MGC59692
81 CDK6/CycD2 CDK6, PLSTIRE
82 CDK6/CycD3 CDK6, PLSTIRE
83 CDK7/CycH/MAT1 CDK7, CAK1, CDKN7, STK1, p39MO15
84 CDK8/CycC CDK8, K35
85 CDK9/CycK CDK9, C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase
86 CDK9/CycT1 CDK9, C-2k, CDC2L4K35, PITALRE, TAK
87 CHK1 CHEK1, n/a
88 CHK2 CHEK2, CDS1, HuCds1, PP1425, RAD53, bA444G7
89 CK1-alpha1 CSNK1A1, CK1, HLCDGP1, PRO2975
90 CK1-delta CSNK1D, HCKID
91 CK1-epsilon CSNK1E, CKIe, HCKIE, MGC10398
92 CK1-gamma1 CSNK1G1
93 CK1-gamma2 CSNK1G2, CK1g2
94 CK1-gamma3 CSNK1G3
95 CK2-alpha1 CSNK2A1, CKII, CK2A1
96 CK2-alpha2 CSNK2A2, n/a
97 CLK1 CLK1, CLK, CLK/STY
98 CLK2 CLK2, MGC61500, clk2, hCLK2
99 CLK3 CLK3, PHCLK3, PHCLK3/152
100 CLK4 CLK4, DKFZp686A20267, CDC-like kinase 4
101 COT MAP3K8, EST, ESTF, TPL2, Tpl-2, c-COT
102 CSF1-R CSF1R, C-FMS, CD115, CSF-1-R, CSFR, FIM2, FMS
103 CSK CSK, n/a
104 DAPK1 DAPK1, n/a
105 DAPK2 DAPK2, DRP-1
106 DAPK3 DAPK3, ZIP, ZIPK
107 DCAMKL2 DCLK2, DCLK, KIAA0369
108 DDR2 N456S DDR2, MIG20a, NTRKR3, TKT, TYRO10
109 DDR2 T654M DDR2, MIG20a, NTRKR3, TKT, TYRO10
110 DDR2 wt DDR2, MIG20a, NTRKR3, TKT, TYRO10
111 DMPK DMPK, DM, DM1, DM1PK, DMK
112 DNA-PK PRKDC, DNAPK, DNPK1, HYRC, HYRC1, XRCC7, p350
113 DYRK1A DYRK1A, DYRK, DYRK1, HP86, MNB, MNBH
114 DYRK1B DYRK1B, MIRK
115 DYRK2 DYRK2
116 DYRK3 DYRK3, DYRK5, RED, REDK
117 DYRK4 DYRK4
118 EEF2K EEF2K, HSU93850, MGC45041, eEF-2K
119 EGF-R d746-750 EGFR, ERBB, mENA, ERBB1
120 EGF-R d747-749/A750P EGFR, ERBB, mENA, ERBB1
121 EGF-R d747-752/P753S EGFR, ERBB, mENA, ERBB1
122 EGF-R d752-759 EGFR, ERBB, mENA, ERBB1
123 EGF-R G719C EGFR, ERBB, mENA, ERBB1
124 EGF-R G719S EGFR, ERBB, mENA, ERBB1
125 EGF-R L858R EGFR, ERBB, ERBB1
126 EGF-R L861Q EGFR, ERBB, mENA, ERBB1
127 EGF-R T790M EGFR, ERBB, ERBB1
128 EGF-R T790M/L858R EGFR, ERBB, ERBB1
129 EGF-R wt EGFR, ERBB, mENA, ERBB1
130 EIF2AK2 EIF2AK2, EIF2AK1, PKR, PRKR
131 EIF2AK3 EIF2AK3, DKFZp781H1925, PEK, PERK, WRS
132 EML4 ALK ALK
133 EML4 ALK F1174L ALK
134 EPHA1 EPHA1, EPH, EPHT, EPHT1
135 EPHA2 EPHA2, ECK
136 EPHA3 EPHA3, ETK, ETK1, EphA3, HEKECK, HEK4, TYRO4
137 EPHA4 EPHA4, HEK8, SEK, TYRO1
138 EPHA5 EPHA5, CEK7, EHK1, EphA5, HEK7, Hek7, TYRO4
139 EPHA6 EPHA6, EHK2, EHK-2, EPA6
140 EPHA7 EPHA7, EHK3, HEK11
141 EPHA8 EPHA8, EEK, EphA8, HEK3, KIAA1459
142 EPHB1 EPHB1, ELK, NET, Hek6, EPHT2
143 EPHB2 EPHB2, DRT, ERK, Hek5, EPHT3, Tyro5
144 EPHB3 EPHB3, ETK2, HEK2, TYRO6
145 EPHB4 EPHB4, HTK, MYK1, TYRO11
146 ERBB2 725YVMA726 ERBB2, CD340, HER2, MLN19, NGL, TKR1
147 ERBB2 wt ERBB2, NEU, NGL, HER2, TKR1, HER-2
148 ERBB4 ERBB4, n/a
149 ERK1 MAPK3, ERT2, HS44KDAP, HUMKER1A, P44ERK1, P44MAPK, PRKM3
150 ERK2 MAPK1, ERK, ERT1, MAPK2, P42MAPK, PRKM1, PRKM2, p38, p40, p41
151 ERK5 MAPK7, BMK1, ERK4, PRKM7
152 ERK7 MAPK15, ERK8, MAPK15
153 FAK aa2-1052 PTK2, FADK, pp125FAK
154 FER FER, TYK3, c-FER, p94-FER
155 FES FES, FPS
156 FGF-R1 V561M FGFR1, FGFR-1, bFGF-R, FLT2, CEK, CD331
157 FGF-R1 wt FGFR1, H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM
158 FGF-R2 FGFR2, FGFR2, BEK, BFR-1, CD332, CEK3, CFD1, ECT1, FGFR-2, JWS, KGFR, KSAM, K-SAM, TK14, TK25
159 FGF-R3 G697C FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
160 FGF-R3 K650E FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
161 FGF-R3 K650M FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
162 FGF-R3 wt FGFR3, ACH, CD333, CEK2, FGFR-3, HSFGFR3EX, JTK4
163 FGF-R4 FGFR4, TKF, JTK2, MGC20292
164 FGR FGR, SRC2, c-fgr, p55c-fgr
165 FLT3 D835Y FLT3, CD135, FLK2, STK-1, STK1
166 FLT3 ITD FLT3, CD135, FLK2, STK-1, STK1
167 FLT3 wt FLT3, CD135, FLK2, STK-1, STK1
168 FRK FRK, GTK, PTK5, RAK
169 FYN wt FYN, SLK, SYN, p59-Fyn
170 FYN Y531F FYN, SLK, SYN, p59-FYN, cFYN
171 GRK2 ADRBK1
172 GRK3 ADRBK2
173 GRK4 GRK4, GPRK2L, GPRK4, GRK4a, IT11
174 GRK5 GRK5
175 GRK6 GRK6
176 GRK7 GRK7
177 GSG2 GSG2, Haspin
178 GSK3-alpha GSK3A
179 GSK3-beta GSK3B, n/a
180 HCK HCK, JTK9
181 HIPK1 HIPK1, KIAA0630, MGC26642, MGC33446, MGC33548, Myak, Nbak2
182 HIPK2 HIPK2, PRO0593
183 HIPK3 HIPK3, ANPK, DYRK6, FIST, FIST3, PKY, YAK1
184 HIPK4 HIPK4, FLJ32818
185 HRI EIF2AK1, HCR
186 IGF1-R IGF1R, JTK13
187 IKK-alpha CHUK, IKBKA, IKK1, IKKA, NFKBIKA, TCF16
188 IKK-beta IKBKB, IKK2, IKKB, NFKBIKB
189 IKK-epsilon IKBKE, IKKE, IKKI, IKK-i, KIAA0151
190 INS-R INSR, n/a
191 INSR-R INSRR, IRR
192 IRAK1 IRAK1, IRAK, Pelle
193 IRAK4 (untagged) IRAK4, REN64, NY-REN-64
194 ITK ITK, EMT 2, LYK 2, PSCTK2 2, IL2-inducible T-cell kinase
195 JAK1 aa583-1154 S729C JAK1, JAK1A, JAK1B, JTK3
196 JAK1 aa583-1154 wt JAK1, JAK1A, JAK1B, JTK3
197 JAK2 JAK2, n/a
198 JAK3 JAK3, JAKL, L-JAK, LJAK
199 JNK1 MAPK8, PRKM8, SAPK1, JNK1-alpha1
200 JNK2 MAPK9, PRKM9, p54aSAPK, JNK2-alpha2
201 JNK3 MAPK10, JNK3A, p54bSAPK
202 KIT A829P KIT, C-Kit, PBT, CD117, SCFR, c-kit
203 KIT D816H KIT, C-Kit, PBT, CD117, SCFR, c-kit
204 KIT D816V KIT, C-Kit, PBT, CD117, SCFR, c-kit
205 KIT T670I KIT, CD117, SCFR, PBT, C-Kit
206 KIT V559D KIT, C-Kit, PBT, CD117, SCFR, c-kit
207 KIT V559D/T670I KIT, C-Kit, PBT, CD117, SCFR, c-kit
208 KIT V559D/V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
209 KIT V560G KIT, C-Kit, PBT, CD117, SCFR, c-kit
210 KIT V654A KIT, C-Kit, PBT, CD117, SCFR, c-kit
211 KIT wt KIT, C-Kit, PBT, CD117, SCFR, c-kit
212 LCK LCK, n/a
213 LIMK1 LIMK1, LIMK
214 LIMK2 LIMK2
215 LRRK2 G2019S LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
216 LRRK2 I2020T LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
217 LRRK2 R1441C LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
218 LRRK2 wt LRRK2, PARK8, ROCO2, FLJ45829, DKFZp434H2111
219 LTK LTK, TYK1
220 LYN LYN, JTK8
221 MAP3K1 MAP3K1, MAPKKK1, MEKK, MEKK1
222 MAP3K10 MAP3K10, MLK2, MST, MEKK10
223 MAP3K11 MAP3K11, MGC17114, MLK-3, PTK1, SPRK
224 MAP3K7/MAP3K7IP1 MAP3K7, TAK1, TGF1a, MEKK7
225 MAP3K9 MAP3K9, MLK1, PRKE1, MEKK9
226 MAP4K2 MAP4K2, BL44, GCK, RAB8IP
227 MAP4K4 MAP4K4, HGK, MEKKK4, NIK
228 MAP4K5 MAP4K5, KHS1, GCKR, KHS, MAPKKKK5
229 MAPKAPK2 MAPKAPK2, n/a
230 MAPKAPK3 MAPKAPK3, 3PK, MAPKAP, MAPKAP3
231 MAPKAPK5 MAPKAPK5, PRAK
232 MARK1 MARK1, KIAA1477
233 MARK2 MARK2, EMK1, MGC99619, PAR-1, ELKL motif kinase 1
234 MARK3 MARK3, CTAK1, KP78, PAR1A
235 MARK4 MARK4, KIAA1860, MARKL1
236 MASTL MASTL, GLW, GREATWALL, GWL, hGWL, MAST-L, THC2
237 MATK MATK, CHK, CTK, DKFZp434N1212, HHYLTK, HYL, Lsk, MGC1708, MGC2101
238 MEK1 F53L MAP2K1, MAP2K1, MAPKK1, MAPKK 1, MKK1, PRKMK1
239 MEK1 wt MAP2K1, MAPKK1, MKK1, PRKMK1
240 MEK2 MAP2K2, MAPKK2, MKK2, PRKMK2
241 MEK5 MAP2K5, MAP2K5, MAPKK5, MKK5, PRKMK5
242 MEKK2 MAP3K2, MAPKKK2, MEKK2B
243 MEKK3 MAP3K3, MAPKKK3, MEK kinase3
244 MELK MELK, PK38
245 MERTK MERTK, MER, MER-PEN, RP38
246 MET D1228H MET, HGFR, RCCP2
247 MET D1228N MET, HGFR, RCCP2
248 MET F1200I MET, HGFR, RCCP2
249 MET M1250T MET, HGFR, RCCP2
250 MET wt MET, HGFR, RCCP2
251 MET Y1230A MET, HGFR, RCCP2
252 MET Y1230C MET, HGFR, RCCP2
253 MET Y1230D MET, HGFR, RCCP2
254 MET Y1230H MET, HGFR, RCCP2
255 MET Y1235D MET, HGFR, RCCP2
256 MINK1 MINK1, B55, YSK2, MAP4K6, ZC3
257 MKK4 MAP2K4, JNKK, JNKK1, MAPKK4, MEK4, PRKMK4, SEK, SERK1
258 MKK6 S207D/T211D MAP2K6, MAPKK6, MEK6, MKK6, PRKMK6, SAPKK3
259 MKK7 MAP2K7, MAPKK7, MEK7, PRKMK7
260 MKNK1 MKNK1, MNK1
261 MKNK2 MKNK2, MNK2, GPRK7
262 MLK4 n/a, KIAA1804
263 MST1 STK4, KRS2, YSK3
264 MST2 STK3, MST-2, KRS1
265 MST3 STK24, MST-3, MST3B, STK3
266 MST4 MST4, MASK
267 mTOR FRAP1, FRAP, FRAP2, RAFT1, RAPT1, rapamycin target protein
268 MUSK MUSK, n/a
269 MYLK MYLK, smMLCK, FLJ12216, KRP, MLCK, MLCK108, MLCK210
270 MYLK2 MYLK2, KMLC, MLCK, skMLCK
271 MYLK3 MYLK3, caMLCK, MLCK2, MYLK2
272 NEK1 NEK1, KIAA1901, NY-REN-55
273 NEK11 NEK11, FLJ23495
274 NEK2 NEK2, NLK1, HsPK21, HsPK 21
275 NEK3 NEK3, HSPK36, MGC29949
276 NEK4 NEK4, NRK2, STK2
277 NEK6 NEK6, SID6-1512
278 NEK7 NEK7, n/a
279 NEK9 NEK9, DKFZp434D0935, MGC16714, NERCC, NERCC1, Nek8
280 NIK MAP3K14, FTDCR1B, HS, HSNIK
281 NLK NLK, n/a
282 NPM1 ALK n/a, n/a
283 NPM1 ALK F1174L n/a, n/a
284 p38-alpha MAPK14, p38-alpha
285 p38-beta MAPK11, p38-beta
286 p38-delta MAPK13, n/a
287 p38-gamma MAPK12, ERK-6, ERK3, ERK5, ERK6, PRKM12, SAPK-3, SAPK3
288 PAK1 PAK1, PAKalpha
289 PAK2 PAK2, PAK65, PAKgamma
290 PAK3 PAK3, CDKN1A, MRX30, OPHN3, PAK3beta, bPAK, hPAK3
291 PAK4 PAK4, n/a
292 PAK6 PAK6, PAK5
293 PAK7 PAK7, KIAA1264, MGC26232
294 PASK PASK, DKFZP434O051, DKFZp686P2031, KIAA0135, PASKIN, STK3
295 PBK PBK, TOPK, SPK, Nori-3, FLJ14385
296 PDGFR-alpha D842V PDGFRA, PDGFR2, CD140a
297 PDGFR-alpha T674I PDGFRA, PDGFR2, CD140a
298 PDGFR-alpha V561D PDGFRA, PDGFR2, CD140a
299 PDGFR-alpha wt PDGFRA, PDGFR2, CD140a
300 PDGFR-beta PDGFRB, JTK12, PDGFR, CD140B, PDGFR1, PDGF-R-beta
301 PDK1 PDPK1, PKB-like
302 PHKG1 PHKG1, PHKg1
303 PHKG2 PHKG2, PHKg2
304 PI4K2A PI4K2A, PI4KII, PIK42A, RP11-548K23.6
305 PI4K2B PI4K2B, PI4KIIB, PI4KII-BETA, PIK42B
306 PI4KB PI4KB, NPIK, pi4K92, PI4K92, PI4Kbeta, PI4KBETA, PI4K-beta, PI4K-BETA, PI4KIIIBETA, PIK4CB
307 PIK3C2A PIK3C2A, CPK, MGC142218, PI3-K-C2A
308 PIK3C2B PIK3C2B, C2-PI3K, PI3K-C2beta
309 PIK3C2G PIK3C2G, PI3K-C2GAMMA, PI3K-C2-gamma
310 PIK3C3 PIK3C3, hVps34, MGC61518, PI3-kinase type 3, PI3K type 3, Vps34, VPS34
311 PIK3CA/PIK3R1 PIK3CA, MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha
312 PIK3CB D1067A/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
313 PIK3CB D1067V/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
314 PIK3CB D1067Y/PIK3R1 P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
315 PIK3CB E1051K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
316 PIK3CB E633K/PIK3R1 PIK3CB, P110BETA, PI3K, PI3KBETA, PI3K-beta, PIK3C1
317 PIK3CB wt/PIK3R1 PIK3CB, PI3K, PI3KBETA, PI3K-beta, PIK3C1, p110-beta
318 PIK3CD/PIK3R1 PIK3CD, p110D, P110DELTA, PI3K, PI3K-delta, p110-delta
319 PIK3CG PIK3CG, p120-PI3K, PI3CG, PI3K, PI3Kgamma, PI3K-gamma, p110-gamma
320 PIM1 PIM1, PIM
321 PIM2 PIM2, n/a
322 PIM3 PIM3, n/a
323 PIP5K1A PIP5K1A, PIP5K1-alpha, PIP5KIalpha, PtdIns(4)P-5-kinase 1 alpha
324 PIP5K1B PIP5K1B, MSS4, PIP5K1-beta, STM7
325 PIP5K1C PIP5K1C, PIP5K1-gamma, PIP5Kgamma, PIP5K-GAMMA, PIPKIg_v4
326 PKA PRKACA, MGC48865, PKA
327 PKC-alpha PRKCA, PKCA, PRKACA, PKC-alpha
328 PKC-beta1 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
329 PKC-beta2 PRKCB1, PKCB, PRKCB, PRKCB2, MGC41878, PKC-beta
330 PKC-delta PRKCD, MAY1, MGC49908, nPKC-delta
331 PKC-epsilon PRKCE, PKCE, nPKC-epsilon
332 PKC-eta PRKCH, PKC-L, PKCL, PRKCL, nPKC-eta
333 PKC-gamma PRKCG, PKCC, PKCG, SCA14, MGC57564
334 PKC-iota PRKCI, PKCI, DXS1179E, MGC26534, nPKC-iota
335 PKC-mu PRKD1, PKD, PKCM, PKC-MU
336 PKC-nu PRKD3, EPK2
337 PKC-theta PRKCQ, PRKCT, nPKC-theta
338 PKC-zeta PRKCZ, PKC2
339 PKC-zeta wt aa184-592 (PKM-zeta) PRKCZ, PKM-zeta, nPKC-zeta, PKC2
340 PKMYT1 PKMYT1, MYT1
341 PKN3 PKN3, PKNbeta, RP11-545E17.1
342 PLK1 PLK1, PLK, STPK13
343 PLK3 PLK3, CNK, FNK, PRK
344 PRK1 PKN1, DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204
345 PRK2 PKN2, PRKCL2, PAK-2
346 PRKD2 PRKD2, PKD2, HSPC187
347 PRKG1 PRKG1, PKG1, CGKI, MGC71944, PGK, PRKG1B, PRKGR1B, cGKIBETA, cGKI-alph
348 PRKG2 PRKG2, PKG2, PRKGR2, cGKII
349 PRKX PRKX, PKX1
350 PYK2 PTK2B, CADTK, CAKB, FADK2, FAK2, PKB, PTK, PYK2, RAFTK, CAK beta
351 RAF1 Y340D/Y341D (untagged) RAF1, c-RAF
352 RET E762Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
353 RET G691S RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
354 RET M918T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
355 RET R749T RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
356 RET R813Q RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
357 RET S891A RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
358 RET V804E RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
359 RET V804L RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
360 RET V804M RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
361 RET wt RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
362 RET Y791F RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
363 RET Y806H RET, CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, RET-ELE1
364 RIPK2 RIPK2, CARD3, CARDIAK, CCK, GIG30, RICK, RIP-2, RIP2
365 RIPK4 RIPK4, ANKK2, ANKRD3, DIK, MGC129992, MGC129993, PKK, RIP4
366 RIPK5 DSTYK, SgK496, SHIK
367 ROCK1 ROCK1, P160ROCK
368 ROCK2 ROCK2, KIAA0619, ROC2
369 RON MST1R, CD136, CDw136, PTK8
370 ROS ROS1, MCF3
371 RPS6KA1 RPS6KA1, RSK3, HU-1, MAPKAPK1A, RSK, RSK1
372 RPS6KA2 RPS6KA2, RSK1, HU-2, MAPKAPK1C, RSK, RSK3
373 RPS6KA3 RPS6KA3, HU-2, HU-3, ISPK-1, MAPKAPK1B, MRX19, RSK, RSK2
374 RPS6KA4 RPS6KA4, MSK2, RSK-B
375 RPS6KA5 RPS6KA5, MSK1, EC 2.7.11, MGC1911, MSPK1, RLPK, RSKL
376 RPS6KA6 RPS6KA6, RSK4
377 S6K RPS6KB1, S6K1, STK14A
378 S6K-beta RPS6KB2, KLS, P70-beta-1, P70-beta-2, S6K-beta2, S6K2, SRK, p70S6Kb
379 SAK PLK4, SAK, STK18
380 SGK1 SGK, n/a
381 SGK2 SGK2, H-SGK2, dJ138B7.2
382 SGK3 SGKL, CISK, SGK2, SGK3
383 SIK1 SIK1, MSK, SNF1LK, SIK, SIK-1, SNF1LK
384 SIK2 SIK2, QIK, SNF1LK2
385 SIK3 SIK3, L19, QSK, SIK-3
386 SLK SLK, KIAA0204, STK2, bA16H23.1, se20-9
387 SNARK NUAK2, DKFZp434J037
388 SNK PLK2, SNK
389 SRC (GST-HIS-tag) SRC, ASV, SRC1, c-SRC, p60-Src
390 SRMS SRMS, C20orf148, SRM, dJ697K14.1
391 SRPK1 SRPK1, SFRSK1
392 SRPK2 SRPK2, SFRSK2
393 STK17A STK17A, DRAK1
394 STK23 SRPK3, MSSK1, MGC102944
395 STK25 STK25, DKFZp686J1430, SOK1, YSK1
396 STK33 STK33
397 STK39 STK39, STLK3, DCHT, SPAK
398 SYK aa1-635 SYK, n/a
399 TAOK2 TAOK2, KIAA0881, MAP3K17, PSK, PSK1, TAO1, TAO2
400 TAOK3 TAOK3, DPK, JIK, MAP3K18, TAO kinase 3
401 TBK1 TBK1, CDC37, HSPCA, HSPCB, IKBKG, NAK, T2K, TANK, TRAF2
402 TEC TEC, PSCTK4
403 TGFB-R1 TGFBR1, ALK5, ACVRLK4
404 TGFB-R2 TGFBR2, HNPCC6, MFS2, RIIC, TGFR-2, TGFbeta-RII
405 TIE2 R849W TEK, VMCM, TIE-2, VMCM1, CD202B
406 TIE2 wt TEK, VMCM, TIE-2, VMCM1, CD202B
407 TIE2 Y1108F TEK, VMCM, TIE-2, VMCM1, CD202B
408 TIE2 Y897S TEK, VMCM, TIE-2, VMCM1, CD202B
409 TLK1 TLK1, PKU-beta, KIAA0137
410 TLK2 TLK2, MGC44450, PKU-ALPHA
411 TNK1 TNK1, n/a
412 TRK-A G667C MTC, TRK1, TRKA
413 TRK-A wt NTRK1, MTC, TRK, TRK1, TRKA
414 TRK-B NTRK2, GP145-TrkB, TRKB, Trk-B
415 TRK-C NTRK3, GP145-TrkC, TRKC, Trk-C
416 TSF1 STK16, KRCT, MPSK, PKL12
417 TSK2 TSSK2, DGS-G, SPOGA2, FLJ38613
418 TSSK1 TSSK1, FKSG81, SPOGA4, STK22D
419 TTBK1 TTBK1, BDTK
420 TTBK2 TTBK2, BDTK, KIAA1855, RP3-330M21.4
421 TTK TTK, ESK, MPS1L1, PYT
422 TXK TXK, BTKL, PSCTK5, PTK4, RLK
423 TYK2 TYK2, JTK1
424 TYRO3 TYRO3, BYK, Brt, Dtk, Sky, Tif
425 VEGF-R1 FLT1, FLT, VEGFR1
426 VEGF-R2 KDR, FLK1, VEGFR, VEGFR2
427 VEGF-R3 FLT4, PCL, VEGFR3
428 VRK1 VRK1, n/a
429 VRK2 VRK2, n/a
430 WEE1 WEE1, WEE1hu
431 WNK1 WNK1, KDP, KIAA0344, PHA2C, PRKWNK1
432 WNK2 WNK2, KIAA1760, NY-CO-43, P/OKcl.13, PRKWNK2, SDCCAG43
433 WNK3 WNK3, KIAA1566, PRKWNK3
434 YES YES, C-YES, HsT441, P61-YES
435 ZAK MLTK, mlklak, AZK
436 ZAP70 ZAP70, SRK, STD, TZK, ZAP-70

Infos in Brief

Kinase Panel

435 kinases, including 87 disease-relevant kinase
mutants and 19 lipid kinases

Assay Technologies

Protein kinases: FlashPlate™-based radiometric assay;
lipid kinases: ADP-Glo™ assay technology (Promega)

ATP Conc

App. ATP-Km for each kinase

Testing Modes

Single concentration measurement or IC50 profiling
(10 conc in semi-log steps)

Cpd Submission

100 x Stock solution in 100% DMSO or
pre-weighed powder (request guidelines)

Report

Detailed report for each project

Turnaround Time

No fixed time slots; first come - first served;
routinely within 10 working days

Info Sheets

Method: Radiometric Assay, Method: ATP-Glo™ Assay, List of ATP-Km

List of Kinases for this Service

PDF