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List of Available Kinases for in vitro Testing Services
For all in vitro testing services offered by ProQinase kinases can be freely chosen from the following list of currently 219 protein kinases:
| No. |
Kinase
Name |
HGNC Name |
... |
No. |
Kinase
Name |
HGNC Name |
| 1 |
ABL1 |
ABL1 |
|
111 |
LYN |
LYN |
| 2 |
ABL1 TI |
ABL1 |
|
112 |
MAP4K4 |
MAP4K4 |
| 3 |
ABL2 |
ABL2 |
|
113 |
MAPKAPK3 |
MAPKAPK3 |
| 4 |
ACK1 |
TNK2 |
|
114 |
MAPKAPK5 |
MAPKAPK5 |
| 5 |
ACV-R1 |
ACVR1 |
|
115 |
MARK1 |
MARK1 |
| 6 |
ACV-R1B |
ACVR1B |
|
116 |
MARK2 |
MARK2 |
| 7 |
AKT1 |
AKT1 |
|
117 |
MARK3 |
MARK3 |
| 8 |
AKT2 |
AKT2 |
|
118 |
MATK |
MATK |
| 9 |
AKT3 |
AKT3 |
|
119 |
MEK1 wt |
MAP2K1 |
| 10 |
ALK |
ALK |
|
120 |
MEK1 SESE |
MAP2K1 |
| 11 |
AMPK-alpha1 fl |
PRKAA1 |
|
121 |
MERTK |
MERTK |
| 12 |
AMPK-alpha1 tr |
PRKAA1 |
|
122 |
MET |
MET |
| 13 |
ARK5 |
NUAK1 |
|
123 |
MINK1 |
MINK1 |
| 14 |
Aurora-A |
STK6 |
|
124 |
MKK6 SDTD |
MAP2K6 |
| 15 |
Aurora-B |
AURKB |
|
125 |
MST1 |
STK4 |
| 16 |
Aurora-C |
AURKC |
|
126 |
MST2 |
STK3 |
| 17 |
AXL |
AXL |
|
127 |
MST3 |
STK24 |
| 18 |
BLK |
BLK |
|
128 |
MST4 |
MST4 |
| 19 |
BMX |
BMX |
|
129 |
MUSK |
MUSK |
| 20 |
B-RAF wt |
BRAF |
|
130 |
MYLK2 |
MYLK2 |
| 21 |
B-RAF VE |
BRAF |
|
131 |
NEK2 |
NEK2 |
| 22 |
BRK |
PTK6 |
|
132 |
NEK3 |
NEK3 |
| 23 |
BTK |
BTK |
|
133 |
NEK6 |
NEK6 |
| 24 |
CAMK2A |
CAMK2A |
|
134 |
NEK7 |
NEK7 |
| 25 |
CDC42BPB |
CDC42BPB |
|
135 |
NIK |
MAP3K14 |
| 26 |
CDC42BPBA |
CDC42BPB |
|
136 |
NLK |
NLK |
| 27 |
CDK1/CycA |
CDC2 |
|
137 |
p38-alpha |
MAPK14 |
| 28 |
CDK1/CycB1 |
CDC2 |
|
138 |
p38-beta |
MAPK11 |
| 29 |
CDK1/CycE |
CDC2 |
|
139 |
p38-gamma |
MAPK12 |
| 30 |
CDK2/CycA |
CDK2 |
|
140 |
PAK1 |
PAK1 |
| 31 |
CDK2/CycE |
CDK2 |
|
141 |
PAK2 |
PAK2 |
| 32 |
CDK3/CycE |
CDK3 |
|
142 |
PAK3 |
PAK3 |
| 33 |
CDK4/CycD1 |
CDK4 |
|
143 |
PAK4 |
PAK4 |
| 34 |
CDK4/CycD3 |
CDK4 |
|
144 |
PAK6 |
PAK6 |
| 35 |
CDK5/p25NCK |
CDK5 |
|
145 |
PAK7 |
PAK7 |
| 36 |
CDK5/p35NCK |
CDK5 |
|
146 |
PASK |
PASK |
| 37 |
CDK6/CycD1 |
CDK6 |
|
147 |
PBK |
PBK |
| 38 |
CDK7/CycH/MAT1 |
CDK7 |
|
148 |
PCTAIRE1 |
PCTK1 |
| 39 |
CDK8/CycC |
CDK8 |
|
149 |
PDGFR-alpha |
PDGFRA |
| 40 |
CDK9/CycT |
CDK9 |
|
150 |
PDGFR-beta |
PDGFRB |
| 41 |
CHK1 |
CHEK1 |
|
151 |
PDK1 |
PDPK1 |
| 42 |
CHK2 |
CHEK2 |
|
152 |
PIM1 |
PIM1 |
| 43 |
CK1-alpha1 |
CSNK1A1 |
|
153 |
PIM2 |
PIM2 |
| 44 |
CK1-delta |
CSNK1D |
|
154 |
PKA |
PRKACA |
| 45 |
CK1-gamma1 |
CSNK1G1 |
|
155 |
PKC-alpha |
PRKCA |
| 46 |
CK1-gamma2 |
CSNK1G2 |
|
156 |
PKC-beta1 |
PRKCB1 |
| 47 |
CK1-gamma3 |
CSNK1G3 |
|
157 |
PKC-beta2 |
PRKCB1 |
| 48 |
CK2-alpha1 |
CSNK2A1 |
|
158 |
PKC-delta |
PRKCD |
| 49 |
CK2-alpha2 |
CSNK2A2 |
|
159 |
PKC-epsilon |
PRKCE |
| 50 |
CLK1 |
CLK1 |
|
160 |
PKC-eta |
PRKCH |
| 51 |
COT |
MAP3K8 |
|
161 |
PKC-gamma |
PRKCG |
| 52 |
CSF1-R |
CSF1R |
|
162 |
PKC-iota |
PRKCI |
| 53 |
CSK |
CSK |
|
163 |
PKC-mu |
PRKD1 |
| 54 |
DAPK1 |
DAPK1 |
|
164 |
PKC-nu |
PRKD3 |
| 55 |
DAPK2 |
DAPK2 |
|
165 |
PKC-theta |
PRKCQ |
| 56 |
DAPK3 |
DAPK3 |
|
166 |
PKC-zeta |
PRKCZ |
| 57 |
DCAMKL2 |
DCLK2 |
|
167 |
PLK1 |
PLK1 |
| 58 |
DMPK |
DMPK |
|
168 |
PLK3 |
PLK3 |
| 59 |
DYRK1A |
DYRK1A |
|
169 |
PRK1 |
PKN1 |
| 60 |
EEF2K |
EEF2K |
|
170 |
PRKG1 |
PRKG1 |
| 61 |
EGF-R |
EGFR |
|
171 |
PRKG2 |
PRKG2 |
| 62 |
EPHA1 |
EPHA1 |
|
172 |
PRKX |
PRKX |
| 63 |
EPHA2 |
EPHA2 |
|
173 |
PYK2 |
PTK2B |
| 64 |
EPHA3 |
EPHA3 |
|
174 |
RAF1 |
RAF1 |
| 65 |
EPHA4 |
EPHA4 |
|
175 |
RET |
RET |
| 66 |
EPHB1 |
EPHB1 |
|
176 |
RIPK2 |
RIPK2 |
| 67 |
EPHB2 |
EPHB2 |
|
177 |
ROCK1 |
ROCK1 |
| 68 |
EPHB3 |
EPHB3 |
|
178 |
ROCK2 |
ROCK2 |
| 69 |
EPHB4 |
EPHB4 |
|
179 |
RON |
MST1R |
| 70 |
ERBB2 |
ERBB2 |
|
180 |
ROS |
ROS1 |
| 71 |
ERBB4 |
ERBB4 |
|
181 |
RPS6KA1 |
RPS6KA1 |
| 72 |
ERK2 |
MAPK1 |
|
182 |
RPS6KA2 |
RPS6KA2 |
| 73 |
FAK fl |
PTK2 |
|
183 |
RPS6KA3 |
RPS6KA3 |
| 74 |
FAK tr |
PTK2 |
|
184 |
RPS6KA4 |
RPS6KA4 |
| 75 |
FER |
FER |
|
185 |
RPS6KA5 |
RPS6KA5 |
| 76 |
FGF-R1 |
FGFR1 |
|
186 |
RPS6KA6 |
RPS6KA6 |
| 77 |
FGF-R1 VM |
FGFR1 |
|
187 |
S6K |
RPS6KB1 |
| 78 |
FGF-R2 |
FGFR2 |
|
188 |
S6K-beta |
RPS6KB2 |
| 79 |
FGF-R3 |
FGFR3 |
|
189 |
SAK |
PLK4 |
| 80 |
FGF-R4 |
FGFR4 |
|
190 |
SGK1 |
SGK |
| 81 |
FGR |
FGR |
|
191 |
SGK2 |
SGK2 |
| 82 |
FLT3 |
FLT3 |
|
192 |
SGK3 |
SGKL |
| 83 |
FLT3 DY |
FLT3 |
|
193 |
SNARK |
NUAK2 |
| 84 |
FRK |
FRK |
|
194 |
SNK |
PLK2 |
| 85 |
FYN |
FYN |
|
195 |
SRC |
SRC |
| 86 |
GRK2 |
ADRBK1 |
|
196 |
SRPK1 |
SRPK1 |
| 87 |
GRK3 |
ADRBK2 |
|
197 |
SRPK2 |
SRPK2 |
| 88 |
GRK4 |
GRK4 |
|
198 |
STK23 |
SRPK3 |
| 89 |
GRK6 |
GRK6 |
|
199 |
STK33 |
STK33 |
| 90 |
GSK3-alpha |
GSK3A |
|
200 |
SYK |
SYK |
| 91 |
GSK3-beta |
GSK3B |
|
201 |
TBK1 |
TBK1 |
| 92 |
HCK |
HCK |
|
202 |
TEC |
TEC |
| 93 |
HIPK1 |
HIPK1 |
|
203 |
TGFB-R1 |
TGFBR1 |
| 94 |
HIPK3 |
HIPK3 |
|
204 |
TIE2 |
TEK |
| 95 |
HRI |
EIF2AK1 |
|
205 |
TRK-A |
NTRK1 |
| 96 |
IGF1-R |
IGF1R |
|
206 |
TRK-B |
NTRK2 |
| 97 |
IKK-alpha |
CHUK |
|
207 |
TRK-C |
NTRK3 |
| 98 |
IKK-beta |
IKBKB |
|
208 |
TSF1 |
STK16 |
| 99 |
IKK-epsilon |
IKBKE |
|
209 |
TSK2 |
TSSK2 |
| 100 |
INS-R |
INSR |
|
210 |
TTK |
TTK |
| 101 |
IRAK1 |
IRAK1 |
|
211 |
TYRO3 |
TYRO3 |
| 102 |
IRAK4 |
IRAK4 |
|
212 |
VEGF-R1 |
FLT1 |
| 103 |
ITK |
ITK |
|
213 |
VEGF-R2 |
KDR |
| 104 |
JAK2* |
JAK2 |
|
214 |
VEGF-R3 |
FLT4 |
| 105 |
JAK3 |
JAK3 |
|
215 |
VRK1 |
VRK1 |
| 106 |
JNK1 |
MAPK8 |
|
216 |
WEE1 |
WEE1 |
| 107 |
JNK3 |
MAPK10 |
|
217 |
WNK3 |
WNK3 |
| 108 |
KIT |
KIT |
|
218 |
YES |
YES |
| 109 |
LCK |
LCK |
|
219 |
ZAP70 |
ZAP70 |
| 110 |
LIMK1 |
LIMK1 |
|
|
|
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* Use of this kinase is
limited by license. More detailed information is available on request from
ProQinase.
Available services:
High-Throughput Screening & Single Point Profiling
IC50-Determination
Single Compound IC50-Profiling with FreeSelect
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